SYNTHETIC ENKEPHALIN ANALOG WITH PROLONGED PARENTERAL AND ORAL ANALGESIC ACTIVITY

被引:382
作者
ROEMER, D
BUESCHER, HH
HILL, RC
PLESS, J
BAUER, W
CARDINAUX, F
CLOSSE, A
HAUSER, D
HUGUENIN, R
机构
[1] SANDOZ LTD,DIV BIOL & MED RES,CH-4002 BASEL,SWITZERLAND
[2] SANDOZ LTD,DIV CHEM RES PHARMACEUT,CH-4002 BASEL,SWITZERLAND
关键词
D O I
10.1038/268547a0
中图分类号
O [数理科学和化学]; P [天文学、地球科学]; Q [生物科学]; N [自然科学总论];
学科分类号
07 ; 0710 ; 09 ;
摘要
引用
收藏
页码:547 / 549
页数:3
相关论文
共 33 条
[1]   ANALGESIA INDUCED INVIVO BY CENTRAL ADMINISTRATION OF ENKEPHALIN IN RAT [J].
BELLUZZI, JD ;
GRANT, N ;
GARSKY, V ;
SARANTAKIS, D ;
WISE, CD ;
STEIN, L .
NATURE, 1976, 260 (5552) :625-626
[2]  
BIRDSALL NJM, 1976, OPIATES ENDOGENOUS O, P19
[3]   ENDORPHINS - PROFOUND BEHAVIORAL-EFFECTS IN RATS SUGGEST NEW ETIOLOGICAL FACTORS IN MENTAL-ILLNESS [J].
BLOOM, F ;
SEGAL, D ;
LING, N ;
GUILLEMIN, R .
SCIENCE, 1976, 194 (4265) :630-632
[4]   DETERMINING THRESHOLDS OF AVERSIVE BRAIN STIMULATION [J].
BOREN, JJ ;
MALIS, JL .
AMERICAN JOURNAL OF PHYSIOLOGY, 1961, 201 (03) :429-&
[5]  
BRADBURY AF, 1976, OPIATES ENDOGENOUS O, P9
[6]   EVIDENCE FOR ANALGESIC ACTIVITY OF ENKEPHALIN IN MOUSE [J].
BUSCHER, HH ;
HILL, RC ;
ROMER, D ;
CARDINAUX, F ;
CLOSSE, A ;
HAUSER, D ;
PLESS, J .
NATURE, 1976, 261 (5559) :423-425
[7]  
D'amour FE, 1941, J PHARMACOL EXP THER, V72, P74
[8]   SELF-ADMINISTRATION OF PSYCHOACTIVE SUBSTANCES BY MONKEY - A MEASURE OF PSYCHOLOGICAL DEPENDENCE [J].
DENEAU, G ;
YANAGITA, T ;
SEEVERS, MH .
PSYCHOPHARMACOLOGIA, 1969, 16 (01) :30-&
[9]  
EDDY NB, 1953, J PHARMACOL EXP THER, V107, P385
[10]   INDUCTION OF EXCESSIVE GROOMING IN RAT BY FRAGMENTS OF LIPOTROPIN [J].
GISPEN, WH ;
WIEGANT, VM ;
BRADBURY, AF ;
HULME, EC ;
SMYTH, DG ;
SNELL, CR ;
DEWIED, D .
NATURE, 1976, 264 (5588) :794-795