AN EFFICIENT SYNTHESIS OF 1-[C-13]-BROMOBENZENE

被引：2

作者：

GELETNEKY, C

BALZER, H

BOCK, W

BERGER, S

机构：

来源：

JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS | 1995年 / 36卷 / 05期

关键词：

C-13; 1-C-13]-BROMOBENZENE; BENZENE RING LABELING;

D O I：

10.1002/jlcr.2580360515

中图分类号：

Q5 [生物化学];

学科分类号：

071010 ; 081704 ;

摘要：

Various routes to functionalized benzenes labelled in position 1 were compared. 1-[C-13]-Bromobenzene has been synthesized in 7 steps with an overall yield of 5.4% from [C-13]-BaCO3, by optimizing the direct transformation of p-nitrophenol into bromobenzene.

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页码：503 / 507

页数：5

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