DEVELOPMENT OF 4-ALKYLPHENYL ARALKYL ETHERS AND RELATED-COMPOUNDS AS POTENT INSECT JUVENILE-HORMONE MIMETICS AND STRUCTURAL ASPECTS OF THEIR ACTIVITY

被引：15

作者：

HAYASHI, T ^{[1
]}

IWAMURA, H ^{[1
]}

FUJITA, T ^{[1
]}

机构：

[1] KYOTO UNIV,FAC AGR,DEPT AGR CHEM,KYOTO 606,JAPAN

来源：

JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY | 1990年 / 38卷 / 10期

关键词：

D O I：

10.1021/jf00100a019

中图分类号：

S [农业科学];

学科分类号：

09 ;

摘要：

We prepared as insect juvenile hormone mimetics 4-alkylphenyl phenylalkyl and phenoxyalkyl ethers and corresponding pyridine derivatives, in which the oxime moiety of the (4-alkylphenoxy)- alkanaldoxime O-ethers we have already developed is replaced by an aromatic function. The activity, examined against Culex pipiens, of the most potent member was comparable to that of the most active JH mimetics so far known. Their structure-activity profiles were compared with those of the previous, nonaromatic ethers, oximes, and related compounds to make the features characteristic to the aromatic function apparent. © 1990, American Chemical Society. All rights reserved.

引用

页码：1965 / 1971

页数：7

共 15 条

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