SELECTIVE AND ENANTIOSPECIFIC ACYLATION OF KAPPA-OPIOID RECEPTORS BY (1S,2S)-TRANS-2-ISOTHIOCYANATO-N-METHYL-N-[2-(1-PYRROLIDINYL)CYCLOHEXYL]BENZENEACETAMIDE - DEMONSTRATION OF KAPPA-RECEPTOR HETEROGENEITY

被引:40
|
作者
DECOSTA, BR
ROTHMAN, RB
BYKOV, V
JACOBSON, AE
RICE, KC
机构
[1] NIDDKD,NEUROSCI LAB,DRUG DESIGN & SYNTH SECT,BETHESDA,MD 20892
[2] NIMH,CLIN STUDIES LAB,RECEPTOR STUDIES UNIT,BETHESDA,MD 20892
关键词
D O I
10.1021/jm00122a001
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
引用
收藏
页码:281 / 283
页数:3
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