THE BETA-ADRENERGIC RADIOLIGAND [H-3] CGP-12177, GENERALLY CLASSIFIED AS AN ANTAGONIST, IS A THERMOGENIC AGONIST IN BROWN ADIPOSE-TISSUE

被引:125
作者
MOHELL, N
DICKER, A
机构
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D O I
10.1042/bj2610401
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
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页码:401 / 405
页数:5
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共 32 条
[1]   ATYPICAL BETA-ADRENOCEPTOR ON BROWN ADIPOCYTES AS TARGET FOR ANTI-OBESITY DRUGS [J].
ARCH, JRS ;
AINSWORTH, AT ;
CAWTHORNE, MA ;
PIERCY, V ;
SENNITT, MV ;
THODY, VE ;
WILSON, C ;
WILSON, S .
NATURE, 1984, 309 (5964) :163-165
[2]   BETA-ADRENERGIC RECEPTORS IN BROWN-ADIPOSE TISSUE - CHARACTERIZATION AND ALTERATIONS DURING ACCLIMATION OF RATS TO COLD [J].
BUKOWIECKI, L ;
FOLLEA, N ;
VALLIERES, J ;
LEBLANC, J .
EUROPEAN JOURNAL OF BIOCHEMISTRY, 1978, 92 (01) :189-196
[3]  
CHENG Y, 1973, BIOCHEM PHARMACOL, V22, P3099
[4]   QUANTITATIVE CONTRIBUTION OF BROWN ADIPOSE-TISSUE THERMOGENESIS TO OVERALL METABOLISM [J].
FOSTER, DO .
CANADIAN JOURNAL OF BIOCHEMISTRY AND CELL BIOLOGY, 1984, 62 (07) :618-622
[5]   SEASONAL CONTROL OF ENERGY-REQUIREMENTS FOR THERMOREGULATION IN THE DJUNGARIAN HAMSTER (PHODOPUS-SUNGORUS), LIVING IN NATURAL PHOTOPERIOD [J].
HELDMAIER, G ;
STEINLECHNER, S .
JOURNAL OF COMPARATIVE PHYSIOLOGY, 1981, 142 (04) :429-437
[6]  
Hemmingsen A. M., 1960, REPORTS STENO MEM HO, V9, P1
[7]   CHARACTERISTICS OF BETA-ADRENERGIC RECEPTORS IN BROWN ADIPOCYTES OF TEMPERATURE-ACCLIMATED RATS [J].
KURAHASHI, M ;
KUROSHIMA, A .
BIOMEDICAL RESEARCH-TOKYO, 1981, 2 (02) :126-133
[8]  
LACASA D, 1986, J LIPID RES, V27, P368
[9]   DIRECT ASSESSMENT OF BETA-ADRENERGIC RECEPTORS IN INTACT RAT ADIPOCYTES BY BINDING OF [H-3]CGP-12177 - EVIDENCE FOR AGONIST HIGH-AFFINITY BINDING COMPLEX AND FOR BETA-1 AND BETA-2 RECEPTOR SUBTYPES [J].
LACASA, D ;
AGLI, B ;
GIUDICELLI, Y .
EUROPEAN JOURNAL OF BIOCHEMISTRY, 1985, 146 (02) :339-346
[10]  
LANG PH, 1985, J CYCLIC NUCL PROT, V10, P341