NEW INDOLE-DERIVATIVES - SYNTHESIS OF 3-ACYL-1-CARBETHOXY-2-TRIFLUOROMETHANESULFONYLINDOLES AND OF SUBSTITUTED 2-VINYLINDOLES

被引：27

作者：

BECCALLI, EM

MARCHESINI, A

机构：

[1] Istituto di Chimica Organica, Facolta' di Farmacia, Universita' degli Studi di Milano, 20133 Milano

来源：

TETRAHEDRON | 1995年 / 51卷 / 08期

关键词：

D O I：

10.1016/0040-4020(94)01092-E

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

3-Acyl-1-carbethoxy-2-trifluoromethanesulfonylindoles 6 and 3-acyl-2-vinylindoles 7 are synthesized from 3-[(1-chloro)alkylidene]indol-2(3H)-ones 2 via 1-carbethoxy-3-[(1-dimethylamino)alkylidene]indol-2(3H)-ones 4.

引用

页码：2353 / 2362

页数：10

共 19 条

[1] STUDIES ON PYRAN DERIVATIVES .91. SYNTHESIS AND PHARMACOLOGICAL TEST OF 2-SUBSTITUTED AND 3-SUBSTITUTED PYRANO [2,3-B] INDOLONES [J].

BARTSCH, H ;

EIDEN, F ;

BUCHBORN, H .

ARCHIV DER PHARMAZIE, 1982, 315 (06) :481-490

[2]

BECCALLI EM, 1994, TETRAHEDRON, V50, P12697

[3] UBER EINE NEUE SYNTHESE DES BETA-OXINDOLYL-(3)-ALANINS (ALPHA-OXY-TRYPTOPHANS) - EIN BEITRAG ZUM ANWENDUNGSBEREICH DER SORENSENSCHEN AMINOSAURE-SYNTHESE [J].

BEHRINGER, H ;

WEISSAUER, H .

CHEMISCHE BERICHTE-RECUEIL, 1952, 85 (7-8) :743-751

[4]

CONWAY SC, 1990, HETEROCYCLES, V30, P627

[5] STUDIES ON THE PREPARATION OF 2-INDOLYL TRIFLATES AND RELATED-COMPOUNDS [J].

CONWAY, SC ;

GRIBBLE, GW .

SYNTHETIC COMMUNICATIONS, 1992, 22 (20) :2987-2995

[6] PALLADIUM-MEDIATED TRANSFORMATIONS OF HETEROAROMATIC TRIFLATES [J].

CRISP, GT ;

PAPADOPOULOS, S .

AUSTRALIAN JOURNAL OF CHEMISTRY, 1989, 42 (02) :279-285

[7] PALLADIUM-CATALYZED CARBONYLATIVE COUPLING OF ARYL TRIFLATES WITH ORGANOSTANNANES [J].

ECHAVARREN, AM ;

STILLE, JK .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1988, 110 (05) :1557-1565

[8] PALLADIUM-CATALYZED COUPLING OF ARYL TRIFLATES WITH ORGANOSTANNANES [J].

ECHAVARREN, AM ;

STILLE, JK .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1987, 109 (18) :5478-5486

[9] PALLADIUM-CATALYZED COUPLING OF 3-INDOLYL TRIFLATE - SYNTHESES OF 3-VINYLINDOLES AND 3-ALKYNYLINDOLES [J].

GRIBBLE, GW ;

CONWAY, SC .

SYNTHETIC COMMUNICATIONS, 1992, 22 (15) :2129-2141

[10]

Horner L, 1941, LIEBIGS ANN CHEM, V548, P117

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