SYNTHESIS AND ANTI-SCHISTOSOMAL ACTIVITY OF CERTAIN PYRAZOLO[1,5-A]PYRIMIDINES

被引：141
作者：
SENGA, K
NOVINSON, T
WILSON, HR
ROBINS, RK
机构：
[1] BRIGHAM YOUNG UNIV,DEPT CHEM,PROVO,UT 84602
[2] ICN PHARMACEUT INC,COVINA,CA 91722
来源：
JOURNAL OF MEDICINAL CHEMISTRY | 1981年 / 24卷 / 05期
关键词：
D O I：
10.1021/jm00137a023
中图分类号：
R914 [药物化学];
学科分类号：
100701 ;
摘要：
引用
收藏
页码：610 / 613
页数：4
相关论文
共 21 条
[1]  
Archer S, 1972, Prog Drug Res, V16, P11
[2]  
CHECCHI S, 1955, GAZZ CHIM ITAL, V85, P1558
[3]   PATHWAYS OF NUCLEOTIDE-METABOLISM IN SCHISTOSOMA-MANSONI .5. ADENOSINE CLEAVAGE ENZYME AND EFFECTS OF PURINE ANALOGS ON ADENOSINE METABOLISM IN-VITRO [J].
CRABTREE, GW ;
SENFT, AW .
BIOCHEMICAL PHARMACOLOGY, 1974, 23 (03) :649-660
[4]   SITES OF ACTION OF ALLOPURINOL IN CRITHIDIA-FASCICULATA [J].
DEWEY, VC ;
KIDDER, GW .
JOURNAL OF PROTOZOOLOGY, 1973, 20 (05) :678-682
[5]   PYRAZOLO[1,5-A]PYRIMIDINES [J].
DORN, H ;
ZUBEK, A .
JOURNAL FUR PRAKTISCHE CHEMIE, 1971, 313 (05) :969-&
[6]   ANTISCHISTOSOMAL ACTION OF TUBERCIDIN ADMINISTERED AFTER ABSORPTION INTO RED CELLS [J].
JAFFE, JJ ;
MEYMARIAN, E ;
DOREMUS, HM .
NATURE, 1971, 230 (5293) :408-+
[7]  
MAKISUMI Y, 1962, CHEM PHARM BULL, V10, P612
[8]   ANTITRYPANOSOMAL EFFECT OF ALLOPURINOL - CONVERSION INVIVO TO AMINOPYRAZOLOPYRIMIDINE NUCLEOTIDES BY TRYPANOSOMA-CRUZI [J].
MARR, JJ ;
BERENS, RL .
SCIENCE, 1978, 201 (4360) :1018-1020
[9]   ANTI-LEISHMANIAL EFFECT OF ALLOPURINOL .2. RELATIONSHIP OF ADENINE METABOLISM IN LEISHMANIA SPECIES TO ACTION OF ALLOPURINOL [J].
MARR, JJ ;
BERENS, RL .
JOURNAL OF INFECTIOUS DISEASES, 1977, 136 (06) :724-732
[10]   3-SUBSTITUTED 5,7-DIMETHYLPYRAZOLO[1,5-A]PYRIMIDINES, 3',5'-CYCLIC-AMP PHOSPHODIESTERASE INHIBITORS .1. [J].
NOVINSON, T ;
HANSON, R ;
DIMMITT, MK ;
SIMON, LN ;
ROBINS, RK ;
OBRIEN, DE .
JOURNAL OF MEDICINAL CHEMISTRY, 1974, 17 (06) :645-648
123