Synthesis and Biological Evaluation of 2-Amino-4H-pyran-3,4,5-tricarboxylate Salt Derivatives

被引:7
作者
Akbari, Ali [1 ]
Azami-Sardooei, Zabihollah [2 ]
Hosseini-Nia, Asghar [3 ]
机构
[1] Univ Jiroft, Fac Sci, Dept Chem, POB 8767161167, Jiroft, Iran
[2] Univ Jiroft, Fac Agr, Dept Corp Protect, Jiroft, Iran
[3] Natl Res Stn Ornamental Plants, Dept Plant Protect, Mahallat, Iran
来源
JOURNAL OF THE KOREAN CHEMICAL SOCIETY-DAEHAN HWAHAK HOE JEE | 2013年 / 57卷 / 04期
关键词
Biological evaluation; Antibacterial activity; 4H-Pyran-3,4,5-tricarboxylate; BF3.SiO2;
D O I
10.5012/jkcs.2013.57.4.455
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
A novel and simple method for the synthesis of 2-amino-4H-pyran-3,4,5-tricarboxylate derivative and the evaluation of their antibacterial activity against Pseudomonas syringae, Xanthomonas citi and Pectobacterium carotovorum are reported. The structure of the isolated compounds has been determined by means of H-1/C-13 NMR and FT-IR Spectroscopy. The reaction of alkyl isocyanides with acetylenic esters in the presence of dimethyl acetone-1,3-dicarboxylate in the present of BF3.SiO2 at ambient temperature. Some of the compound showed significant inhibition to growth of bacteria.
引用
收藏
页码:455 / 460
页数:6
相关论文
共 28 条
[11]  
Li DH, 2007, ARCH PHARM RES, V30, P1051
[12]   NANO-BF3•SIO2: A REUSABLE AND ECO-FRIENDLY CATALYST FOR SYNTHESIS OF QUINOXALINES [J].
Mirjalili, B. B. F. ;
Bamoniri, A. ;
Akbari, A. .
CHEMISTRY OF HETEROCYCLIC COMPOUNDS, 2011, 47 (04) :487-491
[13]   One-Pot Synthesis of 3,4-Dihydropyrimidin-2(1H)-ones (Thiones) Promoted by Nano-BF3•SiO2 [J].
Mirjalili, B. F. ;
Bamoniri, A. ;
Akbari, A. .
JOURNAL OF THE IRANIAN CHEMICAL SOCIETY, 2011, 8 :S135-S140
[14]   BF3•SiO2: an efficient alternative for the synthesis of 14-aryl or alkyl-14H-dibenzo[a,j]xanthenes [J].
Mirjalili, Bi Bi Fatemeh ;
Bamoniri, Abdolhamid ;
Akbari, Ali .
TETRAHEDRON LETTERS, 2008, 49 (45) :6454-6456
[15]  
Mori K, 1998, SYNLETT, P259
[16]   Chemo- and stereoselective reaction between alkyl isocyanides and dimethyl 1,3-acetonedicarbocxylate in the presence of acetylenic esters [J].
Nasiri, Farogh ;
Nazem, Fatemeh ;
Pourdavaie, Kourosh .
MOLECULAR DIVERSITY, 2007, 11 (02) :101-105
[17]   Efficacy of FIT produce wash and chlorine dioxide on pathogen control in fresh potatoes [J].
Park, E. -J. ;
Gray, P. M. ;
Oh, S. -W. ;
Kronenberg, J. ;
Kang, D. -H. .
JOURNAL OF FOOD SCIENCE, 2008, 73 (06) :M278-M282
[18]   Flavonoids as antioxidants [J].
Pietta, PG .
JOURNAL OF NATURAL PRODUCTS, 2000, 63 (07) :1035-1042
[19]  
Rahman AU, 2001, BIOASSAY TECHNIQUES, P14
[20]   BF3•SiO2-catalyzed one-pot synthesis of α-aminophosphonates in ionic liquid and neat conditions [J].
Reddy, Mudumala Veeranarayana ;
Dindulkar, Someshwar D. ;
Jeong, Yeon Tae .
TETRAHEDRON LETTERS, 2011, 52 (37) :4764-4767