Synthesis and Biological Evaluation of 2-Amino-4H-pyran-3,4,5-tricarboxylate Salt Derivatives

被引：7

作者：

Akbari, Ali ^{[1
]}

Azami-Sardooei, Zabihollah ^{[2
]}

Hosseini-Nia, Asghar ^{[3
]}

机构：

[1] Univ Jiroft, Fac Sci, Dept Chem, POB 8767161167, Jiroft, Iran

[2] Univ Jiroft, Fac Agr, Dept Corp Protect, Jiroft, Iran

[3] Natl Res Stn Ornamental Plants, Dept Plant Protect, Mahallat, Iran

来源：

JOURNAL OF THE KOREAN CHEMICAL SOCIETY-DAEHAN HWAHAK HOE JEE | 2013年 / 57卷 / 04期

关键词：

Biological evaluation; Antibacterial activity; 4H-Pyran-3,4,5-tricarboxylate; BF3.SiO2;

D O I：

10.5012/jkcs.2013.57.4.455

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

A novel and simple method for the synthesis of 2-amino-4H-pyran-3,4,5-tricarboxylate derivative and the evaluation of their antibacterial activity against Pseudomonas syringae, Xanthomonas citi and Pectobacterium carotovorum are reported. The structure of the isolated compounds has been determined by means of H-1/C-13 NMR and FT-IR Spectroscopy. The reaction of alkyl isocyanides with acetylenic esters in the presence of dimethyl acetone-1,3-dicarboxylate in the present of BF3.SiO2 at ambient temperature. Some of the compound showed significant inhibition to growth of bacteria.

引用

页码：455 / 460

页数：6

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