Current developments in G-protein-coupled receptors

被引:38
作者
Libert, Frederick [1 ]
Vassart, Gilbert [2 ]
Parmentier, Marc [1 ]
机构
[1] Univ Libre Bruxelles, Fac Med, Inst Rech Interdisciplinaire, B-1070 Brussels, Belgium
[2] Univ Libre Bruxelles, Fac Med, Serv Genet Med, B-1070 Brussels, Belgium
关键词
D O I
10.1016/0955-0674(91)90142-L
中图分类号
Q2 [细胞生物学];
学科分类号
071009 ; 090102 ;
摘要
The rate at which receptors have been cloned has recently increased dramatically - existing families have been extended and new families created. The rapid cloning by homology of 'orphan receptors' has also stimulated the development of a new reverse pharmacology.
引用
收藏
页码:218 / 223
页数:6
相关论文
共 53 条
[1]   DOPAMINE RECEPTOR SUBTYPES - BEYOND THE D1/D2 CLASSIFICATION [J].
ANDERSEN, PH ;
GINGRICH, JA ;
BATES, MD ;
DEARRY, A ;
FALARDEAU, P ;
SENOGLES, SE ;
CARON, MG .
TRENDS IN PHARMACOLOGICAL SCIENCES, 1990, 11 (06) :231-236
[2]   CLONING AND EXPRESSION OF A CDNA-ENCODING AN ENDOTHELIN RECEPTOR [J].
ARAI, H ;
HORI, S ;
ARAMORI, I ;
OHKUBO, H ;
NAKANISHI, S .
NATURE, 1990, 348 (6303) :730-732
[3]   SYNTHESIS AND USE OF A NOVEL N-FORMYL PEPTIDE DERIVATIVE TO ISOLATE A HUMAN N-FORMYL PEPTIDE RECEPTOR CDNA [J].
BOULAY, F ;
TARDIF, M ;
BROUCHON, L ;
VIGNAIS, P .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1990, 168 (03) :1103-1109
[4]   CLONING AND EXPRESSION OF A RAT D2 DOPAMINE RECEPTOR CDNA [J].
BUNZOW, JR ;
VANTOL, HHM ;
GRANDY, DK ;
ALBERT, P ;
SALON, J ;
CHRISTIE, MJ ;
MACHIDA, CA ;
NEVE, KA ;
CIVELLI, O .
NATURE, 1988, 336 (6201) :783-787
[5]   HUMAN CYTOMEGALOVIRUS ENCODES 3 G-PROTEIN-COUPLED RECEPTOR HOMOLOGS [J].
CHEE, MS ;
SATCHWELL, SC ;
PREDDIE, E ;
WESTON, KM ;
BARRELL, BG .
NATURE, 1990, 344 (6268) :774-777
[6]   A 2ND MOLECULAR-FORM OF D2 DOPAMINE RECEPTOR IN RAT AND BOVINE CAUDATE-NUCLEUS [J].
CHIO, CL ;
HESS, GF ;
GRAHAM, RS ;
HUFF, RM .
NATURE, 1990, 343 (6255) :266-269
[7]   PEPTIDES ON PHAGE - A VAST LIBRARY OF PEPTIDES FOR IDENTIFYING LIGANDS [J].
CWIRLA, SE ;
PETERS, EA ;
BARRETT, RW ;
DOWER, WJ .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1990, 87 (16) :6378-6382
[8]   THE DOPAMINE-D2 RECEPTOR - 2 MOLECULAR-FORMS GENERATED BY ALTERNATIVE SPLICING [J].
DALTOSO, R ;
SOMMER, B ;
EWERT, M ;
HERB, A ;
PRITCHETT, DB ;
BACH, A ;
SHIVERS, BD ;
SEEBURG, PH .
EMBO JOURNAL, 1989, 8 (13) :4025-4034
[9]   MOLECULAR-CLONING AND EXPRESSION OF THE GENE FOR A HUMAN D1 DOPAMINE RECEPTOR [J].
DEARRY, A ;
GINGRICH, JA ;
FALARDEAU, P ;
FREMEAU, RT ;
BATES, MD ;
CARON, MG .
NATURE, 1990, 347 (6288) :72-76
[10]   RANDOM PEPTIDE LIBRARIES - A SOURCE OF SPECIFIC PROTEIN-BINDING MOLECULES [J].
DEVLIN, JJ ;
PANGANIBAN, LC ;
DEVLIN, PE .
SCIENCE, 1990, 249 (4967) :404-406