DISPOSITION OF DETIRELIX, A POTENT LUTEINIZING-HORMONE-RELEASING HORMONE ANTAGONIST, IN RATS AND MONKEYS

被引：15

作者：

CHAN, RL ^{[1
]}

HO, W ^{[1
]}

WEBB, AS ^{[1
]}

LAFARGUE, J ^{[1
]}

NERENBERG, CA ^{[1
]}

机构：

[1] SYNTEX RES CORP,DEPT ANALYT & METAB CHEM,PALO ALTO,CA 94304

来源：

PHARMACEUTICAL RESEARCH | 1988年 / 5卷 / 06期

关键词：

D O I：

10.1023/A:1015947325283

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

引用

页码：335 / 340

页数：6

共 23 条

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[4]

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[6]

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[7]

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[8] ANTAGONISTS OF THE LUTEINIZING-HORMONE RELEASING HORMONE WITH PYRIDYL-ALANINES WHICH COMPLETELY INHIBIT OVULATION AT NANOGRAM DOSAGE [J].

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[9] EFFECTS OF AN LH-RELEASING HORMONE ANTAGONIST ON THE SECRETION OF LH, FSH, PROLACTIN AND OVARIAN-STEROIDS AT DIFFERENT STAGES OF THE LUTEAL PHASE IN THE STUMPTAILED MACAQUE (MACACA-ARCTOIDES) [J].

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[10] PHARMACOKINETICS OF GONADOTROPIN-RELEASING HORMONE - COMPARISON OF SUBCUTANEOUS AND INTRAVENOUS ROUTES [J].

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