STRUCTURE-ACTIVITY STUDIES ON INHIBITION OF GABA BINDING TO RAT-BRAIN MEMBRANES BY MUSCIMOL AND RELATED COMPOUNDS

被引：171
作者：
KROGSGAARDLARSEN, P [1 ]
JOHNSTON, GAR [1 ]
机构：
[1] AUSTRALIAN NATL UNIV, DEPT PHARMACOL, CANBERRA 2600, ACT, AUSTRALIA
来源：
JOURNAL OF NEUROCHEMISTRY | 1978年 / 30卷 / 06期
关键词：
D O I：
10.1111/j.1471-4159.1978.tb10469.x
中图分类号：
Q5 [生物化学]; Q7 [分子生物学];
学科分类号：
071010 ; 081704 ;
摘要：
引用
收藏
页码：1377 / 1382
页数：6
相关论文
共 34 条
[1]   EFFECTS OF GABACULINE ON UPTAKE, BINDING AND METABOLISM OF GABA [J].
ALLAN, RD ;
JOHNSTON, GAR ;
TWITCHIN, B .
NEUROSCIENCE LETTERS, 1977, 4 (01) :51-54
[2]   TRANSPORT OF L-PROLINE BY RAT-BRAIN SLICES [J].
BALCAR, VJ ;
JOHNSTON, GAR ;
STEPHANSON, AL .
BRAIN RESEARCH, 1976, 102 (01) :143-151
[3]   INHIBITION OF GABA TRANSAMINASE-ACTIVITY BY 4-AMINOTETROLIC ACID [J].
BEART, PM ;
UHR, ML ;
JOHNSTON, GA .
JOURNAL OF NEUROCHEMISTRY, 1972, 19 (08) :1849-&
[4]   GABA UPTAKE IN RAT-BRAIN SLICES - INHIBITION BY GABA ANALOGS AND BY VARIOUS DRUGS [J].
BEART, PM ;
JOHNSTON, GA .
JOURNAL OF NEUROCHEMISTRY, 1973, 20 (02) :319-324
[5]   COMPETITIVE INHIBITION OF GABA UPTAKE IN RAT-BRAIN SLICES BY SOME GABA ANALOGS OF RESTRICTED CONFORMATION [J].
BEART, PM ;
JOHNSTON, GA ;
UHR, ML .
JOURNAL OF NEUROCHEMISTRY, 1972, 19 (08) :1855-&
[6]   SYNTHESIS OF SOME INDANONES HAVING NITROGEN-CONTAINING SUBSTITUENTS [J].
BERNEY, D ;
JAUNER, T .
HELVETICA CHIMICA ACTA, 1974, 57 (04) :1198-1204
[7]   STRUCTURE OF MUSCIMOL, A GABA ANALOG OF RESTRICTED CONFORMATION [J].
BREHM, L ;
HJEDS, H ;
KROGSGAA.P .
ACTA CHEMICA SCANDINAVICA, 1972, 26 (03) :1298-&
[8]   ORGANIC HYDROXYLAMINE DERIVATIVES .11. STRUCTURAL ANALOGS OF GAMMA-AMINOBUTYRIC ACID (GABA) OF ISOXAZOLE ENOL-BETAINE TYPE - SYNTHESIS AND CRYSTAL-STRUCTURE OF 3-HYDROXY-5-(3-AMINOPROPYL)ISOXAZOLE ZWITTERION [J].
BREHM, L ;
KROGSGAA.P .
ACTA CHEMICA SCANDINAVICA SERIES B-ORGANIC CHEMISTRY AND BIOCHEMISTRY, 1974, B 28 (06) :625-635
[9]   ANTAGONISM BETWEEN BICUCULLINE AND GABA IN CAT BRAIN [J].
CURTIS, DR ;
DUGGAN, AW ;
FELIX, D ;
JOHNSTON, GA ;
MCLENNAN, H .
BRAIN RESEARCH, 1971, 33 (01) :57-&
[10]   THE EXCITATION AND DEPRESSION OF SPINAL NEURONES BY STRUCTURALLY RELATED AMINO ACIDS [J].
CURTIS, DR ;
WATKINS, JC .
JOURNAL OF NEUROCHEMISTRY, 1960, 6 (02) :117-141
1234