GR32191, A HIGHLY POTENT AND SPECIFIC THROMBOXANE A2 RECEPTOR BLOCKING DRUG ON PLATELETS AND VASCULAR AND AIRWAYS SMOOTH-MUSCLE INVITRO

被引:176
作者
LUMLEY, P
WHITE, BP
HUMPHREY, PPA
机构
关键词
D O I
10.1111/j.1476-5381.1989.tb12017.x
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:783 / 794
页数:12
相关论文
共 44 条
[1]   LIGAND-BINDING TO THROMBOXANE RECEPTORS ON HUMAN-PLATELETS - CORRELATION WITH BIOLOGICAL-ACTIVITY [J].
ARMSTRONG, RA ;
JONES, RL ;
WILSON, NH .
BRITISH JOURNAL OF PHARMACOLOGY, 1983, 79 (04) :953-964
[2]   COMPETITIVE ANTAGONISM AT THROMBOXANE RECEPTORS IN HUMAN-PLATELETS [J].
ARMSTRONG, RA ;
JONES, RL ;
PEESAPATI, V ;
WILL, SG ;
WILSON, NH .
BRITISH JOURNAL OF PHARMACOLOGY, 1985, 84 (03) :595-607
[3]   SOME QUANTITATIVE USES OF DRUG ANTAGONISTS [J].
ARUNLAKSHANA, O ;
SCHILD, HO .
BRITISH JOURNAL OF PHARMACOLOGY AND CHEMOTHERAPY, 1959, 14 (01) :48-58
[4]   EFFECTS OF EPOXYMETHANO ANALOGS OF PROSTAGLANDIN ENDOPEROXIDES ON AGGREGATION, ON RELEASE OF 5-HYDROXYTRYPTAMINE AND ON THE METABOLISM OF 3',5'-CYCLIC-AMP AND CYCLIC-GMP IN HUMAN-PLATELETS [J].
BEST, LC ;
MCGUIRE, MB ;
MARTIN, TJ ;
PRESTON, FE ;
RUSSELL, RGG .
BIOCHIMICA ET BIOPHYSICA ACTA, 1979, 583 (03) :344-351
[7]   AH23848 - A THROMBOXANE RECEPTOR BLOCKING DRUG THAT CAN CLARIFY THE PATHOPHYSIOLOGIC ROLE OF THROMBOXANE-A2 [J].
BRITTAIN, RT ;
BOUTAL, L ;
CARTER, MC ;
COLEMAN, RA ;
COLLINGTON, EW ;
GEISOW, SP ;
HALLETT, P ;
HORNBY, EJ ;
HUMPHREY, PPA ;
JACK, D ;
KENNEDY, I ;
LUMLEY, P ;
MCCABE, PJ ;
SKIDMORE, IF ;
THOMAS, M ;
WALLIS, CJ .
CIRCULATION, 1985, 72 (06) :1208-1218
[8]  
BUNDY G L, 1975, Tetrahedron Letters, V24, P1957
[9]  
COLEMAN R A, 1986, British Journal of Pharmacology, V88, p409P
[10]  
COLEMAN R A, 1987, British Journal of Pharmacology, V91, p407P