RUSTING OF THE LOCK AND KEY MODEL FOR PROTEIN-LIGAND BINDING

被引:179
作者
JORGENSEN, WL
机构
关键词
D O I
10.1126/science.1719636
中图分类号
O [数理科学和化学]; P [天文学、地球科学]; Q [生物科学]; N [自然科学总论];
学科分类号
07 ; 0710 ; 09 ;
摘要
引用
收藏
页码:954 / 955
页数:2
相关论文
共 16 条
[1]   3-DIMENSIONAL STRUCTURE OF AN ANTIGEN-ANTIBODY COMPLEX AT 2.8-A RESOLUTION [J].
AMIT, AG ;
MARIUZZA, RA ;
PHILLIPS, SEV ;
POLJAK, RJ .
SCIENCE, 1986, 233 (4765) :747-753
[2]   STRUCTURAL AND FUNCTIONAL-ASPECTS OF DOMAIN MOTIONS IN PROTEINS [J].
BENNETT, WS ;
HUBER, R .
CRC CRITICAL REVIEWS IN BIOCHEMISTRY, 1984, 15 (04) :291-384
[3]   STRUCTURE AND MECHANISM OF CHYMOTRYPSIN [J].
BLOW, DM .
ACCOUNTS OF CHEMICAL RESEARCH, 1976, 9 (04) :145-152
[4]   3-DIMENSIONAL STRUCTURE OF A COMPLEX OF ANTIBODY WITH INFLUENZA-VIRUS NEURAMINIDASE [J].
COLMAN, PM ;
LAVER, WG ;
VARGHESE, JN ;
BAKER, AT ;
TULLOCH, PA ;
AIR, GM ;
WEBSTER, RG .
NATURE, 1987, 326 (6111) :358-363
[6]   MOLECULAR RECOGNITION - CONFORMATIONAL-ANALYSIS OF LIMITED PROTEOLYTIC SITES AND SERINE PROTEINASE PROTEIN INHIBITORS [J].
HUBBARD, SJ ;
CAMPBELL, SF ;
THORNTON, JM .
JOURNAL OF MOLECULAR BIOLOGY, 1991, 220 (02) :507-530
[7]   STRUCTURAL BASIS OF ACTIVATION AND ACTION OF TRYPSIN [J].
HUBER, R ;
BODE, W .
ACCOUNTS OF CHEMICAL RESEARCH, 1978, 11 (03) :114-122
[8]   A COMPETING SALT-BRIDGE SUPPRESSES HELIX FORMATION BY THE ISOLATED C-PEPTIDE CARBOXYLATE OF RIBONUCLEASE-A [J].
KIM, PS ;
BIERZYNSKI, A ;
BALDWIN, RL .
JOURNAL OF MOLECULAR BIOLOGY, 1982, 162 (01) :187-199
[9]   CALCINEURIN IS A COMMON TARGET OF CYCLOPHILIN-CYCLOSPORINE-A AND FKBP-FK506 COMPLEXES [J].
LIU, J ;
FARMER, JD ;
LANE, WS ;
FRIEDMAN, J ;
WEISSMAN, I ;
SCHREIBER, SL .
CELL, 1991, 66 (04) :807-815
[10]   STRUCTURE OF COMPLEX OF SYNTHETIC HIV-1 PROTEASE WITH A SUBSTRATE-BASED INHIBITOR AT 2.3-A RESOLUTION [J].
MILLER, M ;
SCHNEIDER, J ;
SATHYANARAYANA, BK ;
TOTH, MV ;
MARSHALL, GR ;
CLAWSON, L ;
SELK, L ;
KENT, SBH ;
WLODAWER, A .
SCIENCE, 1989, 246 (4934) :1149-1152