KINETIC-ANALYSIS OF THE POSITIVE INOTROPIC ACTION (PIA) OF OUABAIN IN ISOLATED PERFUSED RABBIT HEART - SLOW ONSET OF PIA AND SLOW BINDING TO NA+, K+- ADENOSINE-TRIPHOSPHATASE

被引:8
作者
HARASHIMA, H [1 ]
SUGIYAMA, Y [1 ]
SAWADA, Y [1 ]
SHIGENOBU, K [1 ]
KASUYA, Y [1 ]
IGA, T [1 ]
HANANO, M [1 ]
机构
[1] UNIV TOKYO,FAC PHARMACEUT SCI,BUNKYO KU,TOKYO 113,JAPAN
来源
JOURNAL OF PHARMACOBIO-DYNAMICS | 1988年 / 11卷 / 08期
关键词
D O I
10.1248/bpb1978.11.533
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:533 / 540
页数:8
相关论文
共 21 条
[1]   HIGH-AFFINITY OUABAIN BINDING-SITE AND LOW-DOSE POSITIVE INOTROPIC EFFECT IN RAT MYOCARDIUM [J].
ADAMS, RJ ;
SCHWARTZ, A ;
GRUPP, G ;
GRUPP, I ;
LEE, SW ;
WALLICK, ET ;
POWELL, T ;
TWIST, VW ;
GATHIRAM, P .
NATURE, 1982, 296 (5853) :167-169
[2]  
Akera T, 1978, PHARMACOL REV, V29, P187
[3]  
Brown L, 1984, Basic Res Cardiol, V79 Suppl, P50
[4]  
CCHS HR, 1981, KLIN WOCHENSCHR, V59, P889
[5]  
Fricke U, 1984, Basic Res Cardiol, V79 Suppl, P119
[6]   BINDING-SITES RELATED TO OUABAIN-INDUCED STIMULATION OR INHIBITION OF SODIUM-PUMP [J].
GODFRAIND, T ;
GHYSELBURTON, J .
NATURE, 1977, 265 (5590) :165-166
[7]  
HARASHIMA H, 1987, CHEM PHARM BULL, V35, P2923
[8]  
KOOMEN JM, 1982, ARCH INT PHARMACOD T, V255, P212
[9]   PHARMACOKINETICS OF DIGOXIN - RELATIONSHIP BETWEEN RESPONSE INTENSITY AND PREDICTED COMPARTMENTAL DRUG LEVELS IN MAN [J].
KRAMER, WG ;
KOLIBASH, AJ ;
LEWIS, RP ;
BATHALA, MS ;
VISCONTI, JA ;
REUNING, RH .
JOURNAL OF PHARMACOKINETICS AND BIOPHARMACEUTICS, 1979, 7 (01) :47-61
[10]   ACTIVE-TRANSPORT AND INOTROPIC STATE IN GUINEA-PIG LEFT ATRIUM [J].
LECHAT, P ;
MALLOY, CR ;
SMITH, TW .
CIRCULATION RESEARCH, 1983, 52 (04) :411-422