FREE-RADICAL CYCLIZATIONS LEADING TO 4-MEMBERED RINGS .1. BETA-LACTAM PRODUCTION USING TRIBUTYLTIN HYDRIDE

被引：43

作者：

FREMONT, SL ^{[1
]}

BELLETIRE, JL ^{[1
]}

HO, DM ^{[1
]}

机构：

[1] UNIV CINCINNATI,DEPT CHEM,CINCINNATI,OH 45221

来源：

TETRAHEDRON LETTERS | 1991年 / 32卷 / 21期

关键词：

D O I：

10.1016/S0040-4039(00)79917-5

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Use of HSnBu3 for the reductive cyclization of suitable enamides having a bromide substituent alpha to the carbonyl group affords beta-lactams in good yields.

引用

页码：2335 / 2338

页数：4

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