ENKEPHALIN ANALOGS ELICITING ANALGESIA AFTER INTRAVENOUS-INJECTION

被引:52
作者
DUTTA, AS [1 ]
GORMLEY, JJ [1 ]
HAYWARD, CF [1 ]
MORLEY, JS [1 ]
SHAW, JS [1 ]
STACEY, GJ [1 ]
TURNBULL, MT [1 ]
机构
[1] ICI LTD,DEPT RES,DIV PHARMACEUT,MACCLESFIELD SK10 4TG,CHESHIRE,ENGLAND
关键词
D O I
10.1016/0024-3205(77)90097-2
中图分类号
R-3 [医学研究方法]; R3 [基础医学];
学科分类号
1001 ;
摘要
引用
收藏
页码:559 / 562
页数:4
相关论文
共 13 条
[1]  
BAJUSZ S, 1976, ACTA BIOCHIM BIOPHYS, V11, P305
[2]   SUPERACTIVE ANTINOCICEPTIVE PENTAPEPTIDE, (D-MET2,PRO5), ENKEPHALINAMIDE [J].
BAJUSZ, S ;
RONAI, AZ ;
SZEKELY, JI ;
GRAF, L ;
DUNAIKOVACS, Z ;
BERZETEI, I .
FEBS LETTERS, 1977, 76 (01) :91-92
[3]  
BAXTER MG, 1977, BRIT J PHARMACOL, V59, pP455
[4]   ANALGESIA INDUCED INVIVO BY CENTRAL ADMINISTRATION OF ENKEPHALIN IN RAT [J].
BELLUZZI, JD ;
GRANT, N ;
GARSKY, V ;
SARANTAKIS, D ;
WISE, CD ;
STEIN, L .
NATURE, 1976, 260 (5552) :625-626
[5]   EVIDENCE FOR ANALGESIC ACTIVITY OF ENKEPHALIN IN MOUSE [J].
BUSCHER, HH ;
HILL, RC ;
ROMER, D ;
CARDINAUX, F ;
CLOSSE, A ;
HAUSER, D ;
PLESS, J .
NATURE, 1976, 261 (5559) :423-425
[6]  
EDDY NB, 1953, J PHARMACOL EXP THER, V107, P385
[7]  
GREEBERG R, 1976, NEUROPEPTIDES PHA S1, V5, P151
[8]   KINETIC PARAMETERS OF NARCOTIC AGONISTS AND ANTAGONISTS WITH PARTICULAR REFERENCE TO N-ALLYLNOROXYMORPHONE (NALOXONE) [J].
KOSTERLITZ, HW ;
WATT, AJ .
BRITISH JOURNAL OF PHARMACOLOGY, 1968, 33 (02) :266-+
[9]  
MALICK JB, 1976, PHARMACOLOGIST, V18, P120
[10]   POLYPEPTIDES .11. TETRAZOLE ANALOGUES OF C-TERMINAL TETRAPEPTIDE AMIDE SEQUENCE OF GASTRINS [J].
MORLEY, JS .
JOURNAL OF THE CHEMICAL SOCIETY C-ORGANIC, 1969, (05) :809-&