RACLOPRIDE, A NEW SELECTIVE LIGAND FOR THE DOPAMINE-D2 RECEPTORS

被引:95
作者
HALL, H [1 ]
KOHLER, C [1 ]
GAWELL, L [1 ]
FARDE, L [1 ]
SEDVALL, G [1 ]
机构
[1] KAROLINSKA INST,DEPT PSYCHIAT & PSYCHOL,S-10401 STOCKHOLM 60,SWEDEN
关键词
D O I
10.1016/0278-5846(88)90001-2
中图分类号
R74 [神经病学与精神病学];
学科分类号
摘要
引用
收藏
页码:559 / &
相关论文
共 12 条
[1]   POTENTIAL NEUROLEPTIC AGENTS .4. CHEMISTRY, BEHAVIORAL PHARMACOLOGY, AND INHIBITION OF [H-3] SPIPERONE BINDING OF 3,5-DISUBSTITUTED N-[(1-ETHYL-2-PYRROLIDINYL)METHYL]-6-METHOXYSALICYLAMIDES [J].
DEPAULIS, T ;
KUMAR, Y ;
JOHANSSON, L ;
RAMSBY, S ;
HALL, H ;
SALLEMARK, M ;
ANGEBYMOLLER, K ;
OGREN, SO .
JOURNAL OF MEDICINAL CHEMISTRY, 1986, 29 (01) :61-69
[2]  
FARDE L, 1987, ARCH GEN PSYCHIAT, V44, P671
[3]   SUBSTITUTED BENZAMIDES AS LIGANDS FOR VISUALIZATION OF DOPAMINE RECEPTOR-BINDING IN THE HUMAN-BRAIN BY POSITRON EMISSION TOMOGRAPHY [J].
FARDE, L ;
EHRIN, E ;
ERIKSSON, L ;
GREITZ, T ;
HALL, H ;
HEDSTROM, CG ;
LITTON, JE ;
SEDVALL, G .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1985, 82 (11) :3863-3867
[4]   QUANTITATIVE-ANALYSIS OF D2 DOPAMINE RECEPTOR-BINDING IN THE LIVING HUMAN-BRAIN BY PET [J].
FARDE, L ;
HALL, H ;
EHRIN, E ;
SEDVALL, G .
SCIENCE, 1986, 231 (4735) :258-261
[5]  
FARDE L, 1988, IN PRESS PSYCHOPHARM
[6]  
HALL H, 1986, ACTA PHARMACOL TOX, V58, P368
[7]  
HALL H, 1986, ACTA PHARMACOL TOX, V58, P61
[8]  
HALL H, 1988, IN PRESS J NEURAL TR
[9]   SPECIFIC INVITRO AND INVIVO BINDING OF H-3-RACLOPRIDE - A POTENT SUBSTITUTED BENZAMIDE DRUG WITH HIGH-AFFINITY FOR DOPAMINE D-2 RECEPTORS IN THE RAT-BRAIN [J].
KOHLER, C ;
HALL, H ;
OGREN, SO ;
GAWELL, L .
BIOCHEMICAL PHARMACOLOGY, 1985, 34 (13) :2251-2259
[10]   AUTORADIOGRAPHIC VISUALIZATION OF DOPAMINE D-2 RECEPTORS IN THE MONKEY BRAIN USING THE SELECTIVE BENZAMIDE DRUG [H-3] RACLOPRIDE [J].
KOHLER, C ;
RADESATER, AC .
NEUROSCIENCE LETTERS, 1986, 66 (01) :85-90