INHIBITION OF PHENYLETHANOLAMINE N-METHYLTRANSFERASE BY BENZYLAMINES .2. IN-VITRO AND IN-VIVO STUDIES WITH 2,3-DICHLORO-ALPHA-METHYLBENZYLAMINE

被引：35

作者：

FULLER, RW ^{[1
]}

ROUSH, BW ^{[1
]}

SNODDY, HD ^{[1
]}

MOLLOY, BB ^{[1
]}

机构：

[1] ELI LILLY & CO,LILLY RES LABS,INDIANAPOLIS,IN 46206

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1973年 / 16卷 / 02期

关键词：

D O I：

10.1021/jm00260a004

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：106 / 109

页数：4

共 9 条

[1]

AXELROD J, 1954, J PHARMACOL EXP THER, V110, P315

[2]

DUBNICK B, 1963, J PHARMACOL EXP THER, V140, P85

[3] INHIBITION OF PHENYLETHANOLAMINE N-METHYLTRANSFERASE BY BENZYLAMINES .1. STRUCTURE-ACTIVITY RELATIONSHIPS [J].

FULLER, RW ;

MOLLOY, BB ;

DAY, WA ;

ROUSH, BW ;

MARSH, MM .

JOURNAL OF MEDICINAL CHEMISTRY, 1973, 16 (02) :101-106

[4] A MICROMETHOD FOR ASSAY OF PHENETHANOLAMINE N-METHYL TRANSFERASE [J].

FULLER, RW ;

HUNT, JM .

ANALYTICAL BIOCHEMISTRY, 1966, 16 (02) :349-&

[5]

FULLER RW, 1968, J PHARM PHARMACOL, V20, P157

[6]

GORDON R, 1966, J PHARMACOL EXP THER, V153, P440

[7]

SHORE PA, 1958, J PHARMACOL EXP THER, V122, P295

[8] STATISTICAL ESTIMATIONS IN ENZYME KINETICS [J].

WILKINSON, G .

BIOCHEMICAL JOURNAL, 1961, 80 (02) :324-&

[9] A NEW APPROACH TO ANALYSIS OF INTERATION BETWEEEN MONOAMINE OXIDASE AND ITS SUBSTRATES AND INHIBITORS [J].

ZELLER, EA .

ANNALS OF THE NEW YORK ACADEMY OF SCIENCES, 1963, 107 (03) :811-&

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