IMPROVED SYNTHESIS OF PREFORMED BOC-AMINO-ACID-BRIDGING GROUPS FOR USE IN SOLID-PHASE PEPTIDE-SYNTHESIS

被引：1
|
作者：
CALMES, M [1 ]
CAVELIER, F [1 ]
DAUNIS, J [1 ]
ELYACOUBI, R [1 ]
JACQUIER, R [1 ]
机构：
[1] UNIV MONTPELLIER 2,URA 468,SYNTH & ETUD PHYSICOCHIM AMINOACIDES & PEPTIDES LAB,F-34095 MONTPELLIER 5,FRANCE
来源：
TETRAHEDRON LETTERS | 1990年 / 31卷 / 14期
关键词：
D O I：
10.1016/S0040-4039(00)88900-5
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
Preformed Boc-aminoacid-bridging groups are synthesized by an improved method, using Tmse temporary protection of the starting 4-(halomethyl)phenylacetic acid or bromoacetic acid. © 1990.
引用
收藏
页码：2003 / 2006
页数：4
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