A FACILE CONVERSION OF ARGININE INTO BETA-HOMOARGININE DIPEPTIDES

被引：9

作者：

BASTIAANS, HMM

ALEWIJNSE, AE

VANDERBAAN, JL

OTTENHEIJM, HCJ

机构：

[1] VRIJE UNIV AMSTERDAM,SCHEIKUNDIG LAB,1081 HV AMSTERDAM,NETHERLANDS

[2] NV ORGANON,SCI DEV GRP,5340 BH OSS,NETHERLANDS

来源：

TETRAHEDRON LETTERS | 1994年 / 35卷 / 41期

关键词：

D O I：

10.1016/S0040-4039(00)78368-7

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Irradiation of the arginine derived diazomethyl ketone 2 in the presence of amino esters gives the corresponding beta-homoarginine dipeptide esters 3c-h in 45-76% yield.

引用

页码：7659 / 7660

页数：2

共 5 条

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[5] ASYMMETRIC SYNTHESES OF THE NATURALLY-OCCURRING BETA-AMINO ACIDS, BETA-LYSINE, BETA-LEUCINE AND BETA-PHENYL-BETA-ALANINE VIA NITRONE CYCLOADDITION [J].

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