[METERGOLINE-H-3 - A NEW LIGAND OF SEROTONIN RECEPTORS IN THE RAT-BRAIN

被引:63
作者
HAMON, M [1 ]
MALLAT, M [1 ]
HERBET, A [1 ]
NELSON, DL [1 ]
AUDINOT, M [1 ]
PICHAT, L [1 ]
GLOWINSKI, J [1 ]
机构
[1] CEA,SERV MOLEC MARQUEES,GIF SUR YVETTE,FRANCE
关键词
D O I
10.1111/j.1471-4159.1981.tb01634.x
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:613 / 626
页数:14
相关论文
共 36 条
[1]   DOMPERIDONE-H-3 - SELECTIVE LIGAND FOR DOPAMINE RECEPTORS [J].
BAUDRY, M ;
MARTRES, MP ;
SCHWARTZ, JC .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1979, 308 (03) :231-237
[2]   D-LSD BINDING TO BRAIN HOMOGENATES - POSSIBLE RELATIONSHIP TO SEROTONIN RECEPTORS [J].
BENNETT, JL ;
AGHAJANIAN, GK .
LIFE SCIENCES, 1974, 15 (11) :1935-1944
[3]  
BENNETT JP, 1976, MOL PHARMACOL, V12, P373
[4]   PARADOXICAL DECREASE OF BRAIN 5-HT TURNOVER BY METERGOLINE, A CENTRAL 5-HT RECEPTOR BLOCKER [J].
BOURGOIN, S ;
ARTAUD, F ;
BOCKAERT, J ;
HERY, F ;
GLOWINSKI, J ;
HAMON, M .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1978, 302 (03) :313-321
[5]   SYNAPTIC PLASMA MEMBRANES FROM RAT BRAIN SYNAPTOSOMES - ISOLATION AND PARTIAL CHARACTERIZATION [J].
COTMAN, CW ;
MATTHEWS, DA .
BIOCHIMICA ET BIOPHYSICA ACTA, 1971, 249 (02) :380-+
[6]   DOPAMINE RECEPTOR-BINDING - DIFFERENTIATION OF AGONIST AND ANTAGONIST STATES WITH H-3-DOPAMINE AND HALOPERIDOL-H-3 [J].
CREESE, I ;
BURT, DR ;
SNYDER, SH .
LIFE SCIENCES, 1975, 17 (06) :993-1001
[7]   H-3-SPIROPERIDOL LABELS SEROTONIN RECEPTORS IN RAT CEREBRAL-CORTEX AND HIPPOCAMPUS [J].
CREESE, I ;
SNYDER, SH .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1978, 49 (02) :201-202
[8]  
ENJALBERT A, 1978, MOL PHARMACOL, V14, P11
[9]   ANTAGONISM OF CENTRAL EFFECTS OF TRYPTAMINE AND 5-HYDROXYTRYPTOPHAN BY 1,6-DIMETHYL-8BETA-CARBOBENZYLOXY-AMINOMETHYL-10ALPHA-ERGOLINE - INTERFERENCE WITH AMPHETAMINE AND DOPA [J].
FERRINI, R ;
GLASSER, A .
PSYCHOPHARMACOLOGIA, 1965, 8 (04) :271-&
[10]  
FILLION GMB, 1978, MOL PHARMACOL, V14, P50