TOTAL SYNTHESIS OF OF4949-III AND OF4949-IV - UNUSUAL EFFECTS OF REMOTE SUBSTITUENTS ON THE RATE OF MACROCYCLIZATION REACTIONS

被引:29
作者
BOGER, DL [1 ]
YOHANNES, D [1 ]
机构
[1] PURDUE UNIV,DEPT MED CHEM,W LAFAYETTE,IN 47907
关键词
D O I
10.1016/S0040-4039(01)93447-1
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
引用
收藏
页码:5061 / 5064
页数:4
相关论文
共 22 条
[1]   TERTIARY PHOSPHANE-TETRACHLOROMETHANE, A VERSATILE REAGENT FOR CHLORINATION, DEHYDRATION, AND P-N LINKAGE [J].
APPEL, R .
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION IN ENGLISH, 1975, 14 (12) :801-811
[2]   SELECTIVELY PROTECTED L-DOPA DERIVATIVES - APPLICATION OF THE BENZYLIC HYDROPEROXIDE REARRANGEMENT [J].
BOGER, DL ;
YOHANNES, D .
JOURNAL OF ORGANIC CHEMISTRY, 1987, 52 (23) :5283-5286
[3]  
BOGER DL, 1989, TETRAHEDRON LETT, V30, P2503
[4]   PRACTICAL SYNTHESIS OF CYCLIC-PEPTIDES, WITH AN EXAMPLE OF DEPENDENCE OF CYCLIZATION YIELD UPON LINEAR SEQUENCE [J].
BRADY, SF ;
VARGA, SL ;
FREIDINGER, RM ;
SCHWENK, DA ;
MENDLOWSKI, M ;
HOLLY, FW ;
VEBER, DF .
JOURNAL OF ORGANIC CHEMISTRY, 1979, 44 (18) :3101-3105
[5]   LARGE-SCALE SYNTHESIS OF A CYCLIC HEXAPEPTIDE ANALOG OF SOMATOSTATIN [J].
BRADY, SF ;
FREIDINGER, RM ;
PALEVEDA, WJ ;
COLTON, CD ;
HOMNICK, CF ;
WHITTER, WL ;
CURLEY, P ;
NUTT, RF ;
VEBER, DF .
JOURNAL OF ORGANIC CHEMISTRY, 1987, 52 (05) :764-769
[6]   THE TOTAL SYNTHESES OF THE ISODITYROSINE-DERIVED CYCLIC TRIPEPTIDES OF4949-III AND K-13 - DETERMINATION OF THE ABSOLUTE-CONFIGURATION OF K-13 [J].
EVANS, DA ;
ELLMAN, JA .
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1989, 111 (03) :1063-1072
[8]   THE 1ST TOTAL SYNTHESIS OF DEOXYBOUVARDIN AND RA-VII, NOVEL ANTITUMOR CYCLIC HEXAPEPTIDES [J].
INABA, T ;
UMEZAWA, I ;
YUASA, M ;
INOUE, T ;
MIHASHI, S ;
ITOKAWA, H ;
OGURA, K .
JOURNAL OF ORGANIC CHEMISTRY, 1987, 52 (13) :2957-2958
[9]  
ITOKAWA H, 1984, CHEM PHARM BULL, V32, P284
[10]   BOUVARDIN AND DEOXYBOUVARDIN, ANTI-TUMOR CYCLIC HEXAPEPTIDES FROM BOUVARDIA-TERNIFOLIA (RUBIACEAE) [J].
JOLAD, SD ;
HOFFMANN, JJ ;
TORRANCE, SJ ;
WIEDHOPF, RM ;
COLE, JR ;
ARORA, SK ;
BATES, RB ;
GARGIULO, RL ;
KRIEK, GR .
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1977, 99 (24) :8040-8045