IMPORTANCE OF GENETIC-FACTORS IN THE REGULATION OF DIAZEPAM METABOLISM - RELATIONSHIP TO S-MEPHENYTOIN, BUT NOT DEBRISOQUIN, HYDROXYLATION PHENOTYPE

被引:263
作者
BERTILSSON, L
HENTHORN, TK
SANZ, E
TYBRING, G
SAWE, J
VILLEN, T
机构
关键词
D O I
10.1038/clpt.1989.40
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
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页码:348 / 355
页数:8
相关论文
共 41 条
[11]   DIAZEPAM EFFECTS AND KINETICS IN CAUCASIANS AND ORIENTALS [J].
GHONEIM, MM ;
KORTTILA, K ;
CHIANG, CK ;
JACOBS, L ;
SCHOENWALD, RD ;
MEWALDT, SP ;
KAYABA, KO .
CLINICAL PHARMACOLOGY & THERAPEUTICS, 1981, 29 (06) :749-756
[12]   DIAZEPAM DISPOSITION DETERMINANTS [J].
GREENBLATT, DJ ;
ALLEN, MD ;
HARMATZ, JS ;
SHADER, RI .
CLINICAL PHARMACOLOGY & THERAPEUTICS, 1980, 27 (03) :301-312
[13]   BENZODIAZEPINE KINETICS - IMPLICATIONS FOR THERAPEUTICS AND PHARMACOGERIATRICS [J].
GREENBLATT, DJ ;
DIVOLL, M ;
ABERNETHY, DR ;
OCHS, HR ;
SHADER, RI .
DRUG METABOLISM REVIEWS, 1983, 14 (02) :251-292
[14]  
GREENBLATT DJ, 1981, BR J CLIN PHARM, V1, P35
[15]  
INABA T, 1985, DRUG METAB DISPOS, V13, P443
[16]   PHARMACOKINETIC MODEL FOR DIAZEPAM AND ITS MAJOR METABOLITE DESMETHYLDIAZEPAM FOLLOWING DIAZEPAM ADMINISTRATION [J].
JACK, ML ;
COLBURN, WA .
JOURNAL OF PHARMACEUTICAL SCIENCES, 1983, 72 (11) :1318-1323
[17]   GENETIC-POLYMORPHISM OF MEPHENYTOIN P(4')-HYDROXYLATION - DIFFERENCE BETWEEN ORIENTALS AND CAUCASIANS [J].
JURIMA, M ;
INABA, T ;
KADAR, D ;
KALOW, W .
BRITISH JOURNAL OF CLINICAL PHARMACOLOGY, 1985, 19 (04) :483-487
[18]   THE GENETIC-DEFECT OF MEPHENYTOIN HYDROXYLATION [J].
KALOW, W .
XENOBIOTICA, 1986, 16 (05) :379-389
[19]   ALTERED ELIMINATION OF DESMETHYLDIAZEPAM IN THE ELDERLY [J].
KLOTZ, U ;
MULLERSEYDLITZ, P .
BRITISH JOURNAL OF CLINICAL PHARMACOLOGY, 1979, 7 (01) :119-120
[20]  
KLOTZ U, 1977, CLIN PHARMACOL THER, V21, P430