SUBSTRATES AND INHIBITORS OF ATP-CITRATE LYASE FROM ADIPOSE-TISSUE

被引:0
|
作者
MERSMANN, HJ [1 ]
BROWN, LJ [1 ]
HOUK, JM [1 ]
RAO, DR [1 ]
STEFFEN, DG [1 ]
机构
[1] SHELL DEV CO, BIOL SCI RES CTR, MODESTO, CA 95352 USA
来源
INTERNATIONAL JOURNAL OF BIOCHEMISTRY | 1977年 / 8卷 / 11期
关键词
D O I
10.1016/0020-711X(77)90031-3
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:773 / 779
页数:7
相关论文
共 50 条
  • [1] REGULATION OF ATP-CITRATE LYASE IN RAT ADIPOSE-TISSUE
    RAMAKRISHNA, S
    BENJAMIN, WB
    ANNALS OF THE NEW YORK ACADEMY OF SCIENCES, 1986, 478 : 304 - 306
  • [2] ATP-CITRATE LYASE PHOSPHORYLATION IN RAT ADIPOSE-TISSUE
    PUCCI, DL
    RAMAKRISHNA, S
    BENJAMIN, WB
    JOURNAL OF BIOLOGICAL CHEMISTRY, 1983, 258 (21) : 2907 - 2911
  • [3] ATP CITRATE LYASE IN HUMAN ADIPOSE-TISSUE
    SUZUKI, M
    OKUDA, H
    JOURNAL OF NUTRITIONAL SCIENCE AND VITAMINOLOGY, 1981, 27 (06) : 595 - 598
  • [4] Antimycins, inhibitors of ATP-citrate lyase, from a Streptomyces sp.
    Barrow, CJ
    Oleynek, JJ
    Marinelli, V
    Sun, HH
    Kaplita, P
    Sedlock, DM
    Gillum, AM
    Chadwick, CC
    Cooper, R
    JOURNAL OF ANTIBIOTICS, 1997, 50 (09): : 729 - 733
  • [5] NADPH AND SUBSTRATES PROTECT ATP-CITRATE LYASE FROM THERMAL AND PROTEOLYTIC INACTIVATION
    VOGEL, HJ
    BRIDGER, WA
    JOURNAL OF BIOLOGICAL CHEMISTRY, 1981, 256 (22) : 1702 - 1707
  • [6] EVIDENCE FOR A FUNCTIONAL ATP-CITRATE LYASE - NADP-MALATE DEHYDROGENASE PATHWAY IN BOVINE ADIPOSE-TISSUE - ENZYME AND METABOLITE LEVELS
    SMITH, SB
    PRIOR, RL
    ARCHIVES OF BIOCHEMISTRY AND BIOPHYSICS, 1981, 211 (01) : 192 - 201
  • [7] ATP-citrate lyase deficiency in the mouse
    Beigneux, AP
    Kosinski, C
    Gavino, B
    Horton, JD
    Skarnes, WC
    Young, SG
    JOURNAL OF BIOLOGICAL CHEMISTRY, 2004, 279 (10) : 9557 - 9564
  • [8] ATP-citrate lyase (ACLY) inhibitors as therapeutic agents: a patenting perspective
    Granchi, Carlotta
    EXPERT OPINION ON THERAPEUTIC PATENTS, 2022, 32 (07) : 731 - 742
  • [9] 2-Hydroxy-N-arylbenzenesulfonamides as ATP-citrate lyase inhibitors
    Li, James J.
    Wang, Haixia
    Tino, Joseph A.
    Robl, Jeffrey A.
    Herpin, Timothy F.
    Lawrence, R. Michael
    Biller, Scott
    Jamil, Haris
    Ponticiello, Randy
    Chen, Luping
    Chu, Ching-hsuen
    Flynn, Neil
    Cheng, Dong
    Zhao, Rulin
    Chen, Bangchi
    Schnur, Dora
    Obermeier, Mary T.
    Sasseville, Vito
    Padmanabha, Ramesh
    Pike, Kristen
    Harrity, Thomas
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2007, 17 (11) : 3208 - 3211
  • [10] Design and synthesis of emodin derivatives as novel inhibitors of ATP-citrate lyase
    Koerner, Steffi K.
    Hanai, Jun-Ichi
    Bai, Sha
    Jernigan, Finith E.
    Oki, Miwa
    Komaba, Chieko
    Shuto, Emi
    Sukhatme, Vikas P.
    Sun, Lijun
    EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 126 : 920 - 928