SYNTHESIS AND APPLICATION OF SOME NEW 5-SULFONYL-N-HETEROCYCLO-8-HYDROXYQUINOLINE DERIVATIVES AS POTENTIAL-DRUGS

被引：8

作者：

HAFEZ, AAA ^{[1
]}

AWAD, IMA ^{[1
]}

机构：

[1] UNIV ASSIUT, FAC SCI, DEPT CHEM, ASSIUT, EGYPT

来源：

PHOSPHORUS SULFUR AND SILICON AND THE RELATED ELEMENTS | 1991年 / 61卷 / 3-4期

关键词：

SYNTHESIS; 5-SULFONYL-8-HYDROXYQUINOLINE DERIVATIVES; N-SULFONYL PYRAZOLINES; THEIR CHELATES AND BIOLOGICAL SCREENING;

D O I：

10.1080/10426509108036821

中图分类号：

O61 [无机化学];

学科分类号：

070301 ; 081704 ;

摘要：

Some new sulphonyl-N-heterocyclo-8-hydroxy quinolines have been synthesised by the reaction of 8- hydroxyquinoline-5-sulphonyl hydrazide with different active methylene compounds. The pyrazole, pyrazoline, pyrazolidine and pyridazine derivatives were reacted with some metal cations to give the corresponding chelates. All synthesized compounds have been screened in vitro for their biological activities. © 1991, Taylor & Francis Group, LLC. All rights reserved.

引用

页码：381 / 389

页数：9

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