(+)-1-(3S,4R)-[3-(4-PHENYLBENZYL)-4-HYDROXYCHROMAN-7-YL]CYCLOPENTANE CARBOXYLIC-ACID, A HIGHLY POTENT, SELECTIVE LEUKOTRIENE B-4 ANTAGONIST WITH ORAL ACTIVITY IN THE MURINE COLLAGEN-INDUCED ARTHRITIS MODEL

被引：48

作者：

KOCH, K ^{[1
]}

MELVIN, LS ^{[1
]}

REITER, LA ^{[1
]}

BIGGERS, MS ^{[1
]}

SHOWELL, HJ ^{[1
]}

GRIFFITHS, RJ ^{[1
]}

PETTIPHER, ER ^{[1
]}

CHENG, JB ^{[1
]}

MILICI, AJ ^{[1
]}

BRESLOW, R ^{[1
]}

CONKLYN, MJ ^{[1
]}

SMITH, MA ^{[1
]}

HACKMAN, BC ^{[1
]}

DOHERTY, NS ^{[1
]}

SALTER, E ^{[1
]}

FARRELL, CA ^{[1
]}

SCHULTE, G ^{[1
]}

机构：

[1] PFIZER INC, DIV CENT RES, DEPT IMMUNOL & INFECT DIS, GROTON, CT 06340 USA

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1994年 / 37卷 / 20期

关键词：

D O I：

10.1021/jm00046a001

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

[No abstract available]

引用

页码：3197 / 3199

页数：3

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