SYNTHESIS AND BIOLOGICAL-ACTIVITY OF THE FUNCTIONAL-DERIVATIVES OF 3-(DIMETHYLAMINOMETHYL)-1,2-DITHIOLANES AND 4-(DIMETHYLAMINOMETHYL)-1,2-DITHIOLANES

被引：5
作者：
UNEME, H
MITSUDERA, H
YAMADA, J
KAMIKADO, T
KONO, Y
MANABE, Y
NUMATA, M
机构：
[1] Agricultural Research Laboratories, Agro Division, Takeda Chemical Industries Ltd., Ibaraki 300-42, 10 Wadai, Tsukuba
[2] Department of Medical Entomology, National Institute of Health, Tokyo 141, 2-10-35 Kamiosaki, Shinagawa-ku
来源：
BIOSCIENCE BIOTECHNOLOGY AND BIOCHEMISTRY | 1992年 / 56卷 / 10期
关键词：
D O I：
10.1271/bbb.56.1623
中图分类号：
Q5 [生物化学]; Q7 [分子生物学];
学科分类号：
071010 ; 081704 ;
摘要：
A variety of derivatives of 3- and 4-(dimethylaminomethyl)-1,2-dithiolanes were prepared as their biological equivalents in an analogous way to that for the nereistoxin derivatives. Most of them showed insecticidal and acaricidal activity. High potency against Chilo suppressalis was displayed by S,S'-[2-(dimethylaminomethyl)trimethylene] bis(thiobenzoate), and a broad spectrum of activity was observed for 5-(dimethylaminomethyl)-1,2,3-trithiane. The stereochemistry of the 1,3-dithianes is also discussed.
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页码：1623 / 1631
页数：9
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