SYNTHESIS AND BIOLOGICAL-ACTIVITY OF THE FUNCTIONAL-DERIVATIVES OF 3-(DIMETHYLAMINOMETHYL)-1,2-DITHIOLANES AND 4-(DIMETHYLAMINOMETHYL)-1,2-DITHIOLANES

被引：5
|
作者：
UNEME, H
MITSUDERA, H
YAMADA, J
KAMIKADO, T
KONO, Y
MANABE, Y
NUMATA, M
机构：
[1] Agricultural Research Laboratories, Agro Division, Takeda Chemical Industries Ltd., Ibaraki 300-42, 10 Wadai, Tsukuba
[2] Department of Medical Entomology, National Institute of Health, Tokyo 141, 2-10-35 Kamiosaki, Shinagawa-ku
来源：
BIOSCIENCE BIOTECHNOLOGY AND BIOCHEMISTRY | 1992年 / 56卷 / 10期
关键词：
D O I：
10.1271/bbb.56.1623
中图分类号：
Q5 [生物化学]; Q7 [分子生物学];
学科分类号：
071010 ; 081704 ;
摘要：
A variety of derivatives of 3- and 4-(dimethylaminomethyl)-1,2-dithiolanes were prepared as their biological equivalents in an analogous way to that for the nereistoxin derivatives. Most of them showed insecticidal and acaricidal activity. High potency against Chilo suppressalis was displayed by S,S'-[2-(dimethylaminomethyl)trimethylene] bis(thiobenzoate), and a broad spectrum of activity was observed for 5-(dimethylaminomethyl)-1,2,3-trithiane. The stereochemistry of the 1,3-dithianes is also discussed.
引用
收藏
页码：1623 / 1631
页数：9
相关论文
共 50 条
  • [1] OXIDATION OF 1,2-DITHIOLANES
    LINDBERG, B
    BERGSON, G
    ARKIV FOR KEMI, 1965, 23 (3-4): : 319 - +
  • [2] SYNTHESIS AND BIOLOGICAL-ACTIVITY OF 4-ALKYLTHIO-1,2-DITHIOLANES AND RELATED-COMPOUNDS
    MITSUDERA, H
    KAMIKADO, T
    UNEME, H
    KONO, Y
    AGRICULTURAL AND BIOLOGICAL CHEMISTRY, 1990, 54 (07): : 1719 - 1722
  • [3] SYNTHESIS AND BIOLOGICAL-ACTIVITY OF 1,2-DITHIOLANES AND 1,2-DITHIANES BEARING A NITROGEN-CONTAINING SUBSTITUENT
    UNEME, H
    MITSUDERA, H
    KAMIKADO, T
    KONO, Y
    MANABE, Y
    NUMATA, M
    BIOSCIENCE BIOTECHNOLOGY AND BIOCHEMISTRY, 1992, 56 (12) : 2023 - 2033
  • [4] The Many Ways for Reversible Polymerization of 1,2-Dithiolanes
    Wang, Bang-Sen
    Qu, Da-Hu
    CHEMISTRY LETTERS, 2023, 52 (06) : 496 - 502
  • [5] SYNTHESIS AND THERMAL-STABILITY OF 4-SUBSTITUTED 1,2-DITHIOLANES
    TEUBER, L
    CHRISTOPHERSEN, C
    ACTA CHEMICA SCANDINAVICA SERIES B-ORGANIC CHEMISTRY AND BIOCHEMISTRY, 1988, 42 (09): : 629 - 634
  • [6] REDUCTIVE PHOSPHORYLATION OF 1,2-DITHIOLANES WITH DIALKYL PHOSPHITES
    TAZAKI, M
    NAGAHAMA, S
    TAKAGI, M
    CHEMISTRY LETTERS, 1988, (10) : 1619 - 1622
  • [7] SYNTHESIS AND BIOLOGICAL-ACTIVITY OF 1,3-DITHIOLS, 1,2-DITHIOLANES AND 1,3-DITHIANE-2-THIONES
    KUBOTA, S
    TANIGUCHI, E
    ETO, M
    MAEKAWA, K
    JOURNAL OF THE FACULTY OF AGRICULTURE KYUSHU UNIVERSITY, 1977, 22 (1-2): : 1 - 13
  • [8] Structurally Dynamic Hydrogels Derived from 1,2-Dithiolanes
    Barcan, Gregg A.
    Zhang, Xiangyi
    Waymouth, Robert M.
    JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2015, 137 (17) : 5650 - 5653
  • [9] Synthesis of functional 1,2-dithiolanes from 1,3-bis-tert-butyl thioethers
    Scheutz, Georg M.
    Rowell, Jonathan L.
    Wang, Fu-Sheng
    Abboud, Khalil A.
    Peng, Chi-How
    Sumerlin, Brent S.
    ORGANIC & BIOMOLECULAR CHEMISTRY, 2020, 18 (33) : 6509 - 6513
  • [10] Reaction of polymerization-resistant 1,2-dithiolanes with sulfonium ylides
    Tazaki, M
    Kumakura, M
    Nagahama, S
    Takagi, M
    PHOSPHORUS SULFUR AND SILICON AND THE RELATED ELEMENTS, 1995, 106 (1-4): : 227 - 232
12345