[PROPYL-H-3 BETA-CARBOLINE-3-CARBOXYLATE BINDS SPECIFICALLY TO BRAIN BENZODIAZEPINE RECEPTORS

被引：105
作者：
NIELSEN, M [1 ]
SCHOU, H [1 ]
BRAESTRUP, C [1 ]
机构：
[1] AS FERROSAN, RES LABS, DK-2860 SOEBORG, DENMARK
来源：
JOURNAL OF NEUROCHEMISTRY | 1981年 / 36卷 / 01期
关键词：
D O I：
10.1111/j.1471-4159.1981.tb02404.x
中图分类号：
Q5 [生物化学]; Q7 [分子生物学];
学科分类号：
071010 ; 081704 ;
摘要：
引用
收藏
页码：276 / 285
页数：10
相关论文
共 24 条
[1]   GAS CHROMATOGRAPHIC-MASS SPECTROMETRIC EVIDENCE FOR THE IDENTIFICATION OF 1,2,3,4-TETRAHYDRO-BETA-CARBOLINE AS AN INVIVO CONSTITUENT OF RAT-BRAIN [J].
BARKER, SA ;
HARRISON, RE ;
BROWN, GB ;
CHRISTIAN, ST .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1979, 87 (01) :146-154
[2]   ENHANCEMENT OF DIAZEPAM-H-3 BINDING BY SQ 65,396 - NOVEL ANTI-ANXIETY AGENT [J].
BEER, B ;
KLEPNER, CA ;
LIPPA, AS ;
SQUIRES, RF .
PHARMACOLOGY BIOCHEMISTRY AND BEHAVIOR, 1978, 9 (06) :849-851
[3]   HARMAN IN HUMAN-PLATELETS [J].
BIDDER, TG ;
SHOEMAKER, DW ;
BOETTGER, HG ;
EVANS, M ;
CUMMINS, JT .
LIFE SCIENCES, 1979, 25 (02) :157-164
[4]   PHARMACOLOGICAL CHARACTERIZATION OF BENZODIAZEPINE RECEPTORS IN BRAIN [J].
BRAESTRUP, C ;
SQUIRES, RF .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1978, 48 (03) :263-270
[5]   PARTIAL AGONISTS FOR BRAIN GABA-BENZODIAZEPINE RECEPTOR COMPLEX [J].
BRAESTRUP, C ;
NIELSEN, M ;
KROGSGAARDLARSEN, P ;
FALCH, E .
NATURE, 1979, 280 (5720) :331-333
[6]   URINARY AND BRAIN BETA-CARBOLINE-3-CARBOXYLATES AS POTENT INHIBITORS OF BRAIN BENZODIAZEPINE RECEPTORS [J].
BRAESTRUP, C ;
NIELSEN, M ;
OLSEN, CE .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1980, 77 (04) :2288-2292
[7]   BRAIN SPECIFIC BENZODIAZEPINE RECEPTORS [J].
BRAESTRUP, C ;
SQUIRES, RF .
BRITISH JOURNAL OF PSYCHIATRY, 1978, 133 (SEP) :249-260
[8]   SPECIFIC BENZODIAZEPINE RECEPTORS IN RAT-BRAIN CHARACTERIZED BY HIGH-AFFINITY [DIAZEPAM-H-3] BINDING - (AFFINITY BINDING DIAZEPAM ANXIOLYTIC ACTIVITY BRAIN MEMBRANES REGIONAL DISTRIBUTION) [J].
BRAESTRUP, C ;
SQUIRES, RF .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1977, 74 (09) :3805-3809
[9]  
BRAESTRUP C, 1978, ADV PHARMACOL THER, V7, P173
[10]   INFLUENCE OF GABA RECEPTOR AGONISTS AND ANTAGONISTS ON BINDING OF DIAZEPAM-H-3 TO BENZODIAZEPINE RECEPTOR [J].
BRILEY, MS ;
LANGER, SZ .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1978, 52 (01) :129-132
123