THE SYNTHESIS OF 7-CHLORO-1-METHYL-5-PHENYL-1,3-DIHYDRO-2H-1,4-BENZODIAZEPIN-2-ONE-5-C-14 AND 7-NITRO-1-METHYL-5-(2'-FLUOROPHENYL)-1,3-DIHYDRO-2H-1,4-BENZODIAZEPIN-2-ONE-5-C-14

被引：3

作者：

KAEGI, HH

BURGER, W

BADER, GJ

机构：

来源：

JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS | 1982年 / 19卷 / 02期

关键词：

D O I：

10.1002/jlcr.2580190215

中图分类号：

Q5 [生物化学];

学科分类号：

071010 ; 081704 ;

摘要：

引用

页码：289 / 299

页数：11

共 18 条

[1] NEW RING CLOSURE OF 1,4-BENZODIAZEPINE [J].

BLAZEVIC, N ;

KAIFEZ, F .

JOURNAL OF HETEROCYCLIC CHEMISTRY, 1970, 7 (05) :1173-&

[2]

DZIEWONSKI K, 1935, B INT ACAD POL A SMN, P333

[3]

EILINGSFELD H, 1960, ANGEW CHEM, V72, P840

[4] SOME REACTIONS OF ORTHO-HALOBROMOBENZENES WITH NORMAL-BUTYLLITHIUM [J].

GILMAN, H ;

GORSICH, RD .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1956, 78 (10) :2217-2222

[5] SYNTHESIS OF C-14-LABELED 1,4-BENZODIAZEPINES .2. DIAZEPAM-C-14, DEMETHYLDIAZEPAM-C-14 AND KETAZOLAM-C-14 [J].

HSI, RSP .

JOURNAL OF LABELLED COMPOUNDS, 1974, 10 (03) :389-398

[6] SYNTHESIS OF C-14-LABELED 1,4-BENZODIAZEPINES .3. 2-ALLYLOXY-AMINO-7-CHLORO-5-(2-CHLOROPHENYL)-3H-1,4-BENZODIAZEPINE-2-C-14, 8-CHLORO-1-DIMETHYLAMINO-METHYL-6-PHENYL-4H-S-TRIAZOLO[4,3-A][1,4]BENZODIAZEPINE-3A-C-14, AND 8-CHLORO-2,4-DIHYDRO-2-METHYL-6-PHENYL-1H-S-TRIAZOLO[4,3-A][1,4]BENZODIAZEPIN-1-ONE-3A-14 [J].

HSI, RSP ;

JOHNSON, TD .

JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS, 1976, 12 (04) :613-619

[7]

KAEGI HH, UNPUB

[8] UBER NITRILIUMSALZE .2. EINE NEUE CHINAZOLINSYNTHESE [J].

MEERWEIN, H ;

LAASCH, P ;

MERSCH, R ;

NENTWIG, J .

CHEMISCHE BERICHTE-RECUEIL, 1956, 89 (02) :224-238

[9] SYNTHESIS OF 7-CHLORO-1-[CYCLOPROPYLMETHYL-(METHYLENE-C-14]-5-PHENYL-1H-1,4-BENZODIAZEPIN-2 (3H)-ONE AND 7-CHLORO-1-(CYCLOPROPYLMETHYL)-5-PHENYL-1H-1,4-BENZODIAZEPIN-2 (3H)-ONE-5-C-14 [J].

MERRILL, EJ ;

VERNICE, GG .

JOURNAL OF LABELLED COMPOUNDS, 1971, 7 (01) :89-&

[10]

MURRAY A, 1958, ORGANIC SYNTHESES 1, P86

← 1 2 →