COMPARATIVE BINDING AFFINITIES OF TAMOXIFEN, 4-HYDROXYTAMOXIFEN, AND DESMETHYLTAMOXIFEN FOR ESTROGEN-RECEPTORS ISOLATED FROM HUMAN-BREAST CARCINOMA - CORRELATION WITH BLOOD-LEVELS IN PATIENTS WITH METASTATIC BREAST-CANCER

被引:89
作者
FABIAN, C
TILZER, L
STERNSON, L
机构
[1] UNIV KANSAS,DEPT PHARMACEUT CHEM,LAWRENCE,KS 66045
[2] UNIV KANSAS,MED CTR,DEPT MED,DIV MED ONCOL,KANSAS CITY,KS 66103
[3] UNIV KANSAS,MED CTR,DEPT PATHOL,KANSAS CITY,KS 66103
关键词
D O I
10.1002/bdd.2510020407
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:381 / 390
页数:10
相关论文
共 24 条
  • [1] ADAM H, 1979, BIOCH PHARM, V28, P143
  • [2] SIMPLE COMPUTER-PROGRAM FOR QUANTITATION AND SCATCHARD ANALYSIS OF STEROID RECEPTOR PROTEINS
    AITKEN, SC
    LIPPMAN, ME
    [J]. JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 1977, 8 (01) : 77 - 93
  • [3] CHENG YC, 1976, BIOCH PHARMAC, V22, P3099
  • [4] ESTROGEN RECEPTORS AND ANTAGONISM OF STEROID-HORMONE ACTION
    CLARK, JH
    PECK, EJ
    ANDERSON, JN
    [J]. NATURE, 1974, 251 (5474) : 446 - 448
  • [5] ESTROGEN RECEPTOR - ANTIESTROGEN COMPLEX - ATYPICAL BINDING BY UTERINE NUCLEI AND EFFECTS ON UTERINE GROWTH
    CLARK, JH
    ANDERSON, JN
    PECK, EJ
    [J]. STEROIDS, 1973, 22 (05) : 707 - 718
  • [6] FABIAN C, 1980, CANCER TREAT REP, V64, P765
  • [7] FABIAN C, CANCER
  • [8] METABOLISM OF TAMOXIFEN (ICI 46,474) .2. FEMALE PATIENTS
    FROMSON, JM
    PEARSON, S
    BRAMAH, S
    [J]. XENOBIOTICA, 1973, 3 (11) : 711 - 714
  • [9] ANDROGENS ON ESTROGEN-RECEPTOR .2. CORRELATION BETWEEN NUCLEAR TRANSLOCATION AND UTERINE PROTEIN-SYNTHESIS
    GARCIA, M
    ROCHEFORT, H
    [J]. STEROIDS, 1977, 29 (01) : 111 - 126
  • [10] PAIRED-ION CHROMATOGRAPHIC ANALYSIS OF TAMOXIFEN AND 2 MAJOR METABOLITES IN PLASMA
    GOLANDER, Y
    STERNSON, LA
    [J]. JOURNAL OF CHROMATOGRAPHY, 1980, 181 (01): : 41 - 49