AGONIST VERSUS ANTAGONIST BINDING TO ALPHA-ADRENERGIC RECEPTORS

被引:156
作者
HOFFMAN, BB
MICHEL, T
KILPATRICK, DM
LEFKOWITZ, RJ
TOLBERT, MEM
GILMAN, H
FAIN, JN
机构
[1] DUKE UNIV,MED CTR,HOWARD HUGHES MED RES LAB,DEPT BIOCHEM,DURHAM,NC 27710
[2] BROWN UNIV,PHYSIOL CHEM SECT,PROVIDENCE,RI 02912
来源
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES | 1980年 / 77卷 / 08期
关键词
D O I
10.1073/pnas.77.8.4569
中图分类号
Q [生物科学];
学科分类号
07 ; 0710 ; 09 ;
摘要
引用
收藏
页码:4569 / 4573
页数:5
相关论文
共 27 条
[1]   ADRENERGIC-RECEPTOR OF THE ALPHA1-SUBTYPE MEDIATES THE ACTIVATION OF THE GLYCOGEN-PHOSPHORYLASE IN NORMAL RAT-LIVER [J].
AGGERBECK, M ;
GUELLAEN, G ;
HANOUNE, J .
BIOCHEMICAL PHARMACOLOGY, 1980, 29 (04) :643-645
[2]   FUNCTIONAL BASIS FOR CLASSIFICATION OF ALPHA-ADRENERGIC RECEPTORS [J].
BERTHELSEN, S ;
PETTINGER, WA .
LIFE SCIENCES, 1977, 21 (05) :595-606
[3]  
BIRNBAUM MJ, 1977, J BIOL CHEM, V252, P528
[4]  
CHENG Y, 1973, BIOCHEM PHARMACOL, V22, P3099
[5]  
CLARKE WR, 1978, J BIOL CHEM, V253, P5975
[6]   SIMULTANEOUS ANALYSIS OF FAMILIES OF SIGMOIDAL CURVES - APPLICATION TO BIOASSAY, RADIOLIGAND ASSAY, AND PHYSIOLOGICAL DOSE-RESPONSE CURVES [J].
DELEAN, A ;
MUNSON, PJ ;
RODBARD, D .
AMERICAN JOURNAL OF PHYSIOLOGY, 1978, 235 (02) :E97-E102
[7]   SELECTIVITY OF BLOCKING-AGENTS FOR PRESYNAPTIC AND POSTSYNAPTIC ALPHA-ADRENOCEPTORS [J].
DOXEY, JC ;
SMITH, CFC ;
WALKER, JM .
BRITISH JOURNAL OF PHARMACOLOGY, 1977, 60 (01) :91-96
[8]  
ELREFAI MF, 1979, J BIOL CHEM, V254, P4375
[9]  
EXTON JH, 1979, J CYCLIC NUCL PROT, V5, P277
[10]  
FAIN JN, 1978, RECEPTORS RECOGNIT A, V6, P1