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- [8] IRREVERSIBLE ENZYME INHIBITORS .155. ACTIVE-SITE-DIRECTED IRREVERSIBLE INHIBITORS OF DIHYDROFOLIC REDUCTASE DERIVED FROM 1-[4-(OMEGA-AMINOALKOXY)-3-CHLOROPHENYL]-4,6-DIAMINO-1,2-DIHYDRO-2,2-DIMETHYL-S-TRIAZINES BEARING A TERMINAL SULFONYL FLUORIDE JOURNAL OF MEDICINAL CHEMISTRY, 1969, 12 (04) : 672 - &
- [9] IRREVERSIBLE ENZYME-INHIBITORS .196. ACTIVE-SITE-DIRECTED IRREVERSIBLE INHIBITORS OF DIHYDROFOLATE REDUCTASE DERIVED FROM 1-(4-BENZYLOXY-3-CHLOROPHENYL)-4,6-DIAMINO-1,2-DIHYDRO-2,2-DIMETHYL-S-TRIAZINE AND BEARING A TERMINAL PHENYL SULFONATE GROUP JOURNAL OF MEDICINAL CHEMISTRY, 1972, 15 (09) : 945 - &