STUDY OF KINETICS OF ABSORPTION, DISTRIBUTION AND ELIMINATION OF C-14 N,N-2-DICHLOROETHYL P-AMINO-4, PHENYL BUTYRIC-ACID (CHLORAMINOPHENE) IN RAT

被引:14
作者
GODENECHE, D
MADELMONT, JC
SAUVEZIE, B
BILLAUD, A
机构
[1] INSERM,UNITE RECH ETUD METAB MOLEC MARQUEES,BP 184,63005 CLERMONT FERRAND,FRANCE
[2] CHAIRE THERAPEUTIQUE,30 PL HENRI DUNANT,63003 CLERMONT FERRAND,FRANCE
关键词
D O I
10.1016/0006-2952(75)90342-1
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:1303 / 1308
页数:6
相关论文
共 22 条
[11]   SELECTIVITY OF ACTION OF ALKYLATING AGENTS AND DRUG RESISTANCE .3. UPTAKE AND DEGRADATION OF ALKYLATING DRUGS BY YOSHIDA ASCITES SARCOMA CELLS IN-VITRO [J].
HARRAP, KR ;
HILL, BT .
BIOCHEMICAL PHARMACOLOGY, 1970, 19 (01) :209-&
[13]   ABSORPTION, DISTRIBUTION AND EXCRETION OF H-3-CHLORAMBUCIL IN RATS BEARING YOSHIDA ASCITES SARCOMA [J].
HILL, BT ;
RICHES, PG .
BRITISH JOURNAL OF CANCER, 1971, 25 (04) :831-&
[14]   SELECTIVITY OF ACTION OF ALKYLATING AGENTS AND DRUG RESISTANCE .4. SYNTHESIS OF TRITIUM-LABELED CHLORAMBUCIL AND A STUDY OF ITS CELLULAR UPTAKE BY DRUG-SENSITIVE AND DRUG-RESISTANT STRAINS OF YOSHIDA ASCITES SARCOMA IN-VITRO [J].
HILL, BT ;
JARMAN, M ;
HARRAP, KR .
JOURNAL OF MEDICINAL CHEMISTRY, 1971, 14 (07) :614-&
[15]  
LINFORD JH, 1963, CAN J BIOCHEM PHYS, V41, P931
[16]   ADSORPTION TO HUMAN RED BLOOD CELLS OF CHLORAMBUCIL AND OTHER BIOLOGICAL ALKYLATING AGENTS [J].
LINFORD, JH ;
HRYNIUK, W ;
ISRAELS, LG .
BIOCHEMICAL PHARMACOLOGY, 1969, 18 (12) :2723-&
[17]   RECOVERY OF FREE CHLORAMBUCIL FROM SOLUTION IN BLOOD SERUM [J].
LINFORD, JH .
BIOCHEMICAL PHARMACOLOGY, 1962, 11 (AUG) :693-&
[18]   SYNTHESIS OF C-14-LABELED NN-2-DICHLOROETHYL-4-PARAAMINO PHENYLBUTYRIC ACID (CHLORAMINOPHENE) [J].
MOREAU, J ;
MADELMON.JC .
JOURNAL OF LABELLED COMPOUNDS, 1974, 10 (02) :271-281
[19]   PREPARATION OF TOTAL BLOOD SAMPLES IN VIEW OF C-14 COUNT USING SCINTILLATION IN LIQUID MEDIUM [J].
OUSTRIN, J ;
ROUQUIE, A .
INTERNATIONAL JOURNAL OF APPLIED RADIATION AND ISOTOPES, 1970, 21 (12) :739-&
[20]   STUDIES OF MODE OF ACTION OF TUMOUR-GROWTH-INHIBITING ALKYLATING AGENTS .4. IN-VITRO REACTIONS OF 2-CHLOROETHYLARYLAMINES [J].
ROBERTS, JJ ;
WARWICK, GP .
BIOCHEMICAL PHARMACOLOGY, 1963, 12 (12) :1315-&