Synthesis and antifungal evaluation of imines derived from 3-Amino-2-isopropyl-3H-quinazolin-4-one

被引：0

作者：

Karakaya, Idris ^{[1
,2
]}

Karabuga, Semistan ^{[3
]}

Ulukanli, Zeynep ^{[4
]}

Ulukanli, Sabri ^{[1
]}

机构：

[1] Osmaniye Korkut Ata Univ, Fac Sci & Letters, Dept Chem, Karacaoglan Campus, TR-80000 Osmaniye, Turkey

[2] Ataturk Univ, Fac Sci, Dept Chem, TR-25240 Erzurum, Turkey

[3] Kahramanmaras Sutcu Imam Univ, Fac Sci & Letters, Dept Chem, TR-46100 Kahramanmaras, Turkey

[4] Osmaniye Korkut Ata Univ, Fac Sci & Letters, Dept Biol, TR-80000 Osmaniye, Turkey

来源：

ORGANIC COMMUNICATIONS | 2013年 / 6卷 / 04期

关键词：

Quinazolinone; schiff bases; Imines; antifungal; antimicrobial;

D O I：

暂无

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Novel Schiff bases were synthesised using 3-aminoquinazolinone (1) and a variety of aldehydes in the presence of acetic acid as solvent. Antifungal evaluation of the compounds was carried out by the agar dilution method. Among the all compounds prepared, quinazolinone itself showed the best fungiostatic activity against all filamentous fungi.

引用

页码：139 / 147

页数：9

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