SYNTHESIS AND EVALUATION OF NOVEL ALKYLPIPERAZINES AS POTENTIAL DOPAMINE ANTAGONISTS

被引：14

作者：

GLENNON, RA ^{[1
]}

SALLEY, JJ ^{[1
]}

STEINSLAND, OS ^{[1
]}

NELSON, S ^{[1
]}

机构：

[1] UNIV TEXAS, MED BRANCH, DEPT PHARMACOL & TOXICOL, GALVESTON, TX 77550 USA

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1981年 / 24卷 / 06期

关键词：

D O I：

10.1021/jm00138a007

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：678 / 683

页数：6

共 36 条

[1] EFFECT OF CLOZAPINE ON TURNOVER OF DOPAMINE IN CORPUS STRIATUM AND IN LIMBIC SYSTEM [J].

ANDEN, N ;

STOCK, G .

JOURNAL OF PHARMACY AND PHARMACOLOGY, 1973, 25 (04) :346-348

[2] SYNTHESIS OF PHENANTHRENES .4. 8-CHLORO-4A-METHYL-1,2,3,4,4A,9,10,10A-OCTAHYDROPHENANTHRENE [J].

BARNES, RA ;

KONORT, MD .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1953, 75 (02) :303-305

[3] SYNTHESIS OF TERTIARY ARYLALKYLAMINES FROM ARYL GRIGNARD REAGENTS [J].

BAVIN, PMG ;

GANELLIN, CR ;

LOYNES, JM ;

MILES, PD ;

RIDLEY, HF .

JOURNAL OF MEDICINAL CHEMISTRY, 1966, 9 (05) :790-&

[4] STRUCTURE OF CATECHOLAMINES .2. CRYSTAL STRUCTURE OF DOPAMINE HYDROCHLORIDE [J].

BERGIN, R ;

CARLSTROM, D .

ACTA CRYSTALLOGRAPHICA SECTION B-STRUCTURAL CRYSTALLOGRAPHY AND CRYSTAL CHEMISTRY, 1968, B 24 :1506-+

[5] HOMOCYCLIC RING CLOSURES VIA BENZYNE INTERMEDIATES - A NEW SYNTHESIS OF 1-SUBSTITUTED BENZOCYCLOBUTENES [J].

BUNNETT, JF ;

SKORCZ, JA .

JOURNAL OF ORGANIC CHEMISTRY, 1962, 27 (11) :3836-&

[6]

BURT DR, 1976, MOL PHARMACOL, V12, P800

[7]

CALDWELL AG, 1962, Patent No. 1139504

[8] RIGID CONGENERS OF DOPAMINE BASED ON OCTAHYDROBENZO[F]QUINOLINE - PERIPHERAL AND CENTRAL EFFECTS [J].

CANNON, JG ;

SUAREZGUTIERREZ, C ;

LEE, T ;

LONG, JP ;

COSTALL, B ;

FORTUNE, DH ;

NAYLOR, RJ .

JOURNAL OF MEDICINAL CHEMISTRY, 1979, 22 (04) :341-347

[9] CEREBRAL DOPAMINE AGONIST PROPERTIES OF SOME 2-AMINOTETRALIN DERIVATIVES AFTER PERIPHERAL AND INTRACEREBRAL ADMINISTRATION [J].

CANNON, JG ;

LEE, T ;

GOLDMAN, HD ;

COSTALL, B ;

NAYLOR, RJ .

JOURNAL OF MEDICINAL CHEMISTRY, 1977, 20 (09) :1111-1116

[10]

CARLSSON A, 1978, BIOL PSYCHIAT, V13, P3

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