IDENTIFICATION OF A NEW METABOLITE OF TAMOXIFEN IN PATIENT SERUM DURING BREAST-CANCER THERAPY

被引:20
作者
BAIN, RR [1 ]
JORDAN, VC [1 ]
机构
[1] UNIV WISCONSIN, CTR HLTH SCI, DEPT HUMAN ONCOL, MADISON, WI 53792 USA
关键词
D O I
10.1016/0006-2952(83)90571-3
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:373 / 375
页数:3
相关论文
共 12 条
  • [1] METABOLISM OF TAMOXIFEN IN HUMANS
    ADAM, HK
    DOUGLAS, EJ
    KEMP, JV
    [J]. BIOCHEMICAL PHARMACOLOGY, 1979, 28 (01) : 145 - 147
  • [2] BROWN R, J CHROMAT
  • [3] COEZY E, 1982, CANCER RES, V42, P317
  • [4] DETERMINATION OF TAMOXIFEN AND AN HYDROXYLATED METABOLITE IN PLASMA FROM PATIENTS WITH ADVANCED BREAST-CANCER USING GAS CHROMATOGRAPHY-MASS SPECTROMETRY
    DANIEL, CP
    GASKELL, SJ
    BISHOP, H
    NICHOLSON, RI
    [J]. JOURNAL OF ENDOCRINOLOGY, 1979, 83 (03) : 401 - 408
  • [5] COMPARATIVE BINDING AFFINITIES OF TAMOXIFEN, 4-HYDROXYTAMOXIFEN, AND DESMETHYLTAMOXIFEN FOR ESTROGEN-RECEPTORS ISOLATED FROM HUMAN-BREAST CARCINOMA - CORRELATION WITH BLOOD-LEVELS IN PATIENTS WITH METASTATIC BREAST-CANCER
    FABIAN, C
    TILZER, L
    STERNSON, L
    [J]. BIOPHARMACEUTICS & DRUG DISPOSITION, 1981, 2 (04) : 381 - 390
  • [6] FABIAN C, 1980, CANCER TREAT REP, V64, P765
  • [7] METABOLISM OF TAMOXIFEN (ICI 46,474) .2. FEMALE PATIENTS
    FROMSON, JM
    PEARSON, S
    BRAMAH, S
    [J]. XENOBIOTICA, 1973, 3 (11) : 711 - 714
  • [8] MONOHYDROXYLATED METABOLITE OF TAMOXIFEN WITH POTENT ANTI-ESTROGENIC ACTIVITY
    JORDAN, VC
    COLLINS, MM
    ROWSBY, L
    PRESTWICH, G
    [J]. JOURNAL OF ENDOCRINOLOGY, 1977, 75 (02) : 305 - 316
  • [9] STUDIES ON MECHANISM OF ACTION OF NONSTEROIDAL ANTIOESTROGEN TAMOXIFEN (ICI 46,474) IN RAT
    JORDAN, VC
    DIX, CJ
    ROWSBY, L
    PRESTWICH, G
    [J]. MOLECULAR AND CELLULAR ENDOCRINOLOGY, 1977, 7 (02) : 177 - 192
  • [10] LIPPMAN M, 1976, CANCER RES, V36, P4595