2-STEP SYNTHESIS OF SUBSTITUTED INDOLO[1,2-A]-QUINOXALIN-6-ONES

被引：20

作者：

BEACH, MJ ^{[1
]}

HOPE, R ^{[1
]}

KLAUBERT, DH ^{[1
]}

RUSSELL, RK ^{[1
]}

机构：

[1] RW JOHNSON PHARMACEUT RES INST,RARITAN,NJ 08869

来源：

SYNTHETIC COMMUNICATIONS | 1995年 / 25卷 / 14期

关键词：

D O I：

10.1080/00397919508015898

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The reaction of indole-2-carboxylates with 2-fluoronitrobenzenes in 1-methyl-2-pyrrolidinone containing NaH affords the 1-(2-nitrophenyl)indole-2-carboxlyates 1. These compounds are reduced with iron in acetic acid to afford the indolo[1,2-a]quinoxalin-6(5H)-ones 2.

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页码：2165 / 2183

页数：19

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