SOME NOVEL INHIBITORS OF PORCINE PANCREATIC ELASTASE

被引：37
作者：
HASSALL, CH
JOHNSON, WH
ROBERTS, NA
机构：
[1] Roche Products Limited, Welwyn Garden City, Herts
来源：
BIOORGANIC CHEMISTRY | 1979年 / 8卷 / 03期
关键词：
D O I：
10.1016/0045-2068(79)90057-9
中图分类号：
Q5 [生物化学]; Q7 [分子生物学];
学科分类号：
071010 ; 081704 ;
摘要：
New evidence has enabled the identification of novel specific inhibitors of porcine pancreatic elastase with potential for action in vivo. The basis for optimization of activity in this series of derivatives of alanylproline, and the relationship of elastase inhibition to the binding mode, is discussed. © 1979.
引用
收藏
页码：299 / 309
页数：11
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