A SHORT AND EFFICIENT SYNTHESIS OF 4,5-DIARYLPYRIMIDINES

被引：0
作者：
DOMINGUEZ, E
DEMARIGORTA, EM
OLIVERA, R
SANMARTIN, R
机构：
来源：
SYNLETT | 1995年 / 09期
关键词：
PYRIMIDINE; AMINE EXCHANGE; LEUCKART; ENAMINONE; DEOXYBENZOIN;
D O I：
暂无
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
4,5-Diarylpyrimidines 3 are efficiently prepared by submmiting enaminones 2, readily obtained from deoxybenzoins 1, to Leuckart reaction conditions. This conversion implies an uncommon amine group exchange.
引用
收藏
页码：955 / &
相关论文
共 21 条
  • [1] (E)-3-DIMETHYLAMINO-1,2-DIPHENYL-2-PROPEN-1-ONE - STRUCTURE OF AN ENAMINONE
    ARRIORTUA, MI
    URTIAGA, MK
    DOMINGUEZ, E
    IGARTUA, A
    IRIONDO, C
    SOLANS, X
    [J]. ACTA CRYSTALLOGRAPHICA SECTION C-CRYSTAL STRUCTURE COMMUNICATIONS, 1992, 48 : 528 - 530
  • [2] UBER DIE DARSTELLUNG SUBSTITUIERTER PYRIMIDINE, ISOXAZOLE UND PYRAZOLE
    BREDERECK, H
    HERLINGER, H
    SCHWEIZER, EH
    [J]. CHEMISCHE BERICHTE-RECUEIL, 1960, 93 (05): : 1208 - 1211
  • [3] SAUREAMID-REAKTIONEN .33. TRISACYLAMINOMETHANE - SYNTHESEN UND UMSETZUNGEN
    BREDERECK, H
    EFFENBERGER, F
    TREIBER, HJ
    [J]. CHEMISCHE BERICHTE-RECUEIL, 1963, 96 (06): : 1505 - &
  • [4] Brown Daniel R.L., 2009, IACR CRYPTOL EPRINT, V2009, P620
  • [5] BROWN DJ, 1982, MED RES REV, V2, P191
  • [6] BROWN DJ, 1970, PYRIMIDINES S, V1
  • [7] Brown DJ, 1984, COMPREHENSIVE HETERO, V3, P57
  • [8] ONE-POT SYNTHESIS OF RUFLOXACIN
    CECCHETTI, V
    FRAVOLINI, A
    SCHIAFFELLA, F
    [J]. SYNTHETIC COMMUNICATIONS, 1991, 21 (22) : 2301 - 2308
  • [9] COHN WE, 1963, PROGR NUCLEIC ACID R, V1
  • [10] DOMINGUEZ E, 1984, HETEROCYCLES, V22, P1271
123